SCHEMBL9633071

SCHEMBL9633071

CCCC(=O)c1cc2ccccc2[nH]1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 4/20 0.62
FLT3 P36888 1/20 0.61
KDM4E B2RXH2 3/20 0.59
HPGD P15428 2/20 0.59
MAPT P10636 1/20 0.59
DAO P14920 1/20 0.59
SRD5A2 P31213 1/20 0.59
HSD17B10 Q99714 1/20 0.59
DRD2 P14416 2/20 0.58
DRD3 P35462 1/20 0.58
PDGFRB P09619 3/20 0.58
PDGFRA P16234 3/20 0.58
GAA P10253 2/20 0.57
ALDH1A1 P00352 1/20 0.57
MAPK1 P28482 1/20 0.57
MAOB P27338 1/20 0.54
LMNA P02545 1/20 0.53
TP53 P04637 1/20 0.53
L3MBTL1 Q9Y468 1/20 0.53
HRH4 Q9H3N8 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4454538 0.89 DRD2 (0.62) IDO1FLT3KDM4EHPGDMAPT
SCHEMBL30148093 0.86 IDO1 (0.66) IDO1FLT3KDM4EHPGDMAPT
SCHEMBL2730199 0.86 IDO1 (0.66) IDO1FLT3KDM4EHPGDMAPT
SCHEMBL9100296 0.85 IDO1 (0.64) IDO1FLT3KDM4EHPGDMAPT
SCHEMBL28038704 0.84 IDO1 (0.59) IDO1FLT3KDM4EHPGDMAPT
Indole-2-Carboxylic Acid SCHEMBL30748205 0.83 KDM4E (0.73) IDO1FLT3KDM4EHPGDMAPT
Acetic Acid SCHEMBL11542600 0.82 IDO1 (0.65) IDO1FLT3KDM4EHPGDMAPT
Butyric Acid SCHEMBL28840260 0.81 KDM4E (0.57) IDO1FLT3KDM4EHPGDMAPT
SCHEMBL6923977 0.81 IDO1 (0.68) IDO1FLT3KDM4EHPGDMAPT
SCHEMBL9666519 0.80 IDO1 (0.62) IDO1FLT3KDM4EHPGDMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8377981-B2 CBI derivatives subject to reductive activation THE SCRIPPS RESEARCH INSTITUTE (US) 2013-02-19 US disclosed
US-5089497-A Dopaminergic agents WARNER-LAMBERT COMPANY (US) 1992-02-18 US disclosed
US-4997844-A Compounds for the treatment of allergic or inflammatory diseases or shock conditions ICI AMERICAS INC. (US) 1991-03-05 US disclosed
EP-0179619-B1 HETEROCYCLIC AMIDES ICI AMERICAS INC. (US) 1990-09-05 EP disclosed
EP-0179619-A1 Heterocyclic amides ICI AMERICAS INC. (US) 1986-04-30 EP disclosed