SCHEMBL9635535

SCHEMBL9635535

CCCOC(=O)c1cc(=O)c2cc(O)ccc2o1

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 7/20 0.72
AKR1B1 P15121 4/20 0.64
ALOX15 P16050 2/20 0.52
MAOA P21397 1/20 0.49
ATM Q13315 1/20 0.48
KMT2A Q03164 2/20 0.48
ALDH1A1 P00352 2/20 0.47
ESR1 P03372 1/20 0.47
CHRM1 P11229 1/20 0.47
TSHR P16473 1/20 0.47
SLC6A2 P23975 1/20 0.47
KDR P35968 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
HPGD P15428 2/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
MEN1 O00255 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP2D6 P10635 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29495358 0.89 AKR1B1 (0.80) MAOBAKR1B1ALOX15MAOAKMT2A
SCHEMBL115442 0.89 AKR1B1 (0.80) MAOBAKR1B1ALOX15MAOAKMT2A
SCHEMBL4258065 0.87 MAOB (0.72) MAOBAKR1B1ATMKMT2AALDH1A1
SCHEMBL4251638 0.82 MAOB (0.65) MAOBAKR1B1MAOAATMKMT2A
SCHEMBL2814301 0.80 AKR1B1 (0.69) MAOBAKR1B1ALOX15KMT2AALDH1A1
SCHEMBL4258027 0.80 MAOB (0.62) MAOBAKR1B1ATMKMT2AALDH1A1
SCHEMBL4249673 0.79 MAOB (0.72) MAOBAKR1B1ATMKMT2AALDH1A1
SCHEMBL4254462 0.79 MAOB (0.60) MAOBAKR1B1ALOX15KMT2AALDH1A1
SCHEMBL29495537 0.78 AKR1B1 (1.00) MAOBAKR1B1ALOX15MAOAATM
SCHEMBL1021783 0.78 AKR1B1 (1.00) MAOBAKR1B1ALOX15MAOAATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5082849-A Antiinflammatory agents or antiallergens AVENTIS PHARMACEUTICALS INC. 1992-01-21 US disclosed
EP-0434827-A4 QUINOLINYL-BENZOPYRAN DERIVATIVES AS ANTAGONISTS OF LEUKOTRIENE D 4? 1992-01-08 EP disclosed
EP-0434827-A1 QUINOLINYL-BENZOPYRAN DERIVATIVES AS ANTAGONISTS OF LEUKOTRIENE D 4? RORER INTERNATIONAL (HOLDINGS), INC. (US) 1991-07-03 EP disclosed
WO-1991001123-A2 QUINOLINYL-BENZOPYRAN DERIVATIVES AS ANTAGONISTS OF LEUKOTRIENE D¿4? RORER INTERNATIONAL (OVERSEAS) INC. (US) 1991-02-07 WO disclosed
US-4977162-A Quinolinyl-chromone derivatives and use for treatment of hypersensitive ailments RORER PHARMACEUTICAL CORPORATION (US) 1990-12-11 US disclosed