SCHEMBL9638641

SCHEMBL9638641

NC(=O)c1snc(O)c1Br

nearest known ligand 0.33

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CDC7 O00311 1/20 0.33
DBF4 Q9UBU7 1/20 0.33
GAA P10253 1/20 0.30
ALOX15 P16050 1/20 0.30
MAPK1 P28482 1/20 0.30
HSD17B10 Q99714 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9637680 0.69 IKBKB (0.37) GAAALOX15MAPK1HSD17B10
SCHEMBL8182444 0.67
SCHEMBL11005034 0.66 KDR (0.35) MAPK1
SCHEMBL5497435 0.62
SCHEMBL11559950 0.62
SCHEMBL11792477 0.61 POLB (0.38) GAAMAPK1HSD17B10
SCHEMBL17871026 0.61 GPR35 (0.36)
SCHEMBL27816571 0.60 IKBKB (0.41) CDC7GAAALOX15MAPK1HSD17B10
SCHEMBL626686 0.59 GAA (0.35) CDC7DBF4GAAALOX15MAPK1
SCHEMBL22082145 0.57

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5171860-A Diamino isothiazole-1-oxides and 1,1 dioxides as gastric secretion inhibitors MERCK & CO., INC. (US) 1992-12-15 US disclosed
EP-0067436-B1 DIAMINO ISOTHIAZOLE -1-OXIDES AND -1,1-DIOXIDES AS GASTRIC SECRETION INHIBITORS MERCK & CO. INC. (US) 1986-07-23 EP disclosed
EP-0067436-A2 Diamino isothiazole -1-oxides and -1,1-dioxides as gastric secretion inhibitors MERCK & CO. INC. (US) 1982-12-22 EP disclosed