SCHEMBL9640561

SCHEMBL9640561

CCOc1cc(OCC)nc(NC(C)=O)n1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 3/20 0.66
MAPK8 P45983 2/20 0.55
ADORA3 P0DMS8 5/20 0.48
ADORA2A P29274 1/20 0.48
ALDH1A1 P00352 1/20 0.46
TDP1 Q9NUW8 2/20 0.46
MEN1 O00255 1/20 0.46
LMNA P02545 1/20 0.46
KMT2A Q03164 1/20 0.46
ADORA1 P30542 2/20 0.46
RORC P51449 1/20 0.43
PRKD3 O94806 1/20 0.43
MAP4K4 O95819 1/20 0.43
MAPK9 P45984 1/20 0.43
MAPK10 P53779 1/20 0.43
MAP4K2 Q12851 1/20 0.43
PKN2 Q16513 1/20 0.43
PRKD2 Q9BZL6 1/20 0.43
STK17A Q9UEE5 1/20 0.43
CYP2C9 P11712 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9640545 0.79 CYP1A2 (1.00) CYP1A2ADORA3ALDH1A1KMT2AADORA1
SCHEMBL10397625 0.77 KMT2A (0.43) CYP1A2MAPK8ALDH1A1TDP1MEN1
SCHEMBL9737603 0.77 SMN1; SMN2 (0.40) CYP1A2MAPK8ADORA3ADORA2AALDH1A1
SCHEMBL2986990 0.76 KMT2A (0.50) CYP1A2ALDH1A1MEN1KMT2AMAPT
SCHEMBL15058379 0.76 TSHR (0.44) CYP1A2MAPK8ADORA3ADORA2AALDH1A1
SCHEMBL15305693 0.74 CYP1A2 (0.80) CYP1A2MAPK8ADORA3ALDH1A1MAPK9
SCHEMBL2798552 0.73 MAP2K7 (0.41) CYP1A2MAPK8ADORA3ADORA2AADORA1
SCHEMBL1719546 0.73 MAPK8 (0.41) CYP1A2MAPK8ADORA3ADORA2AALDH1A1
SCHEMBL9505994 0.72 CYP1A2 (0.57) CYP1A2ADORA3ALDH1A1MEN1LMNA
SCHEMBL24271910 0.71 MAPK8 (1.00) CYP1A2MAPK8ADORA3ADORA2ATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0279366-B1 PROCESS FOR THE PREPARATION OF PYRIMIDINES HOECHST AKTIENGESELLSCHAFT (DE) 1992-08-12 EP disclosed
US-4960887-A REACTING PROPANEDIIMIDATE WITH CARBONIC ACID IMINEDERIVATIVE HOECHST AKTIENGESELLSCHAFT (DE) 1990-10-02 US disclosed
EP-0279366-A2 Process for the preparation of pyrimidines HOECHST AKTIENGESELLSCHAFT (DE) 1988-08-24 EP disclosed