SCHEMBL9642008

SCHEMBL9642008

O=c1oc2ccccc2c(O)c1[C@@H]1Cc2ccccc2[C@@H](c2ccc(-c3ccc(Br)cc3)cc2)C1

nearest known ligand 0.85

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
VKORC1 Q9BQB6 2/20 0.85
THRB P10828 1/20 0.42
HTR2A P28223 2/20 0.42
HTR2C P28335 2/20 0.42
HTR2B P41595 2/20 0.42
HRH3 Q9Y5N1 2/20 0.42
NQO1 P15559 2/20 0.41
TP53 P04637 1/20 0.39
TNKS O95271 1/20 0.38
LMNA P02545 1/20 0.38
HPGD P15428 1/20 0.38
TOP2A P11388 1/20 0.38
PRNP P04156 1/20 0.37
RXFP1 Q9HBX9 1/20 0.37
CTSK P43235 1/20 0.36
CYP2C9 P11712 2/20 0.36
KDM4E B2RXH2 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9640911 1.00 VKORC1 (0.85) VKORC1THRBHTR2AHTR2CHTR2B
SCHEMBL9641963 1.00 VKORC1 (0.85) VKORC1THRBHTR2AHTR2CHTR2B
SCHEMBL9642577 1.00 VKORC1 (0.85) VKORC1THRBHTR2AHTR2CHTR2B
SCHEMBL10644371 0.93 VKORC1 (0.73) VKORC1NQO1TP53LMNAHPGD
Brodifacoum SCHEMBL29455095 0.92 VKORC1 (1.00) VKORC1THRBHTR2AHTR2CHTR2B
Brodifacoum SCHEMBL435133 0.92 VKORC1 (1.00) VKORC1THRBHTR2AHTR2CHTR2B
SCHEMBL10688149 0.87 VKORC1 (0.89) VKORC1THRBNQO1TP53TNKS
SCHEMBL25202475 0.86 VKORC1 (0.82) VKORC1THRBNQO1TNKSLMNA
SCHEMBL29904783 0.85 VKORC1 (0.86) VKORC1NQO1TP53LMNAHPGD
SCHEMBL24003588 0.85 VKORC1 (0.86) VKORC1NQO1TP53LMNAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0147052-B1 RODENTICIDES IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1992-09-09 EP disclosed
US-4783481-A TRANS ISOMER OF 3-SUBSTITUTED-4-HYDROXYCOUMARIN IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1988-11-08 US disclosed
EP-0147052-A2 Rodenticides IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1985-07-03 EP disclosed