SCHEMBL9643179

SCHEMBL9643179

CN(C(=O)Cc1ccc(Cl)c(Cl)c1)[C@@H]1c2ccccc2C[C@H]1N1CCCC1

nearest known ligand 0.82

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRK1 P41145 8/20 0.82
SIGMAR1 Q99720 7/20 0.82
OPRM1 P35372 5/20 0.82
OPRD1 P41143 5/20 0.82
CYP3A4 P08684 3/20 0.63
CYP2D6 P10635 3/20 0.63
TP53 P04637 2/20 0.63
TSHR P16473 2/20 0.63
ALDH1A1 P00352 2/20 0.63
MEN1 O00255 1/20 0.63
CYP1A2 P05177 1/20 0.63
CYP2C19 P33261 1/20 0.63
MTOR P42345 1/20 0.63
RAB9A P51151 1/20 0.63
KMT2A Q03164 1/20 0.63
MAPK8 P45983 1/20 0.63
MAPK9 P45984 1/20 0.63
MAPK10 P53779 1/20 0.63
PMP22 Q01453 3/20 0.62
SMN1; SMN2 Q16637 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7962880 1.00 OPRK1 (0.82) OPRK1SIGMAR1OPRM1OPRD1CYP3A4
SCHEMBL7963740 0.99 OPRK1 (0.81) OPRK1SIGMAR1OPRM1OPRD1CYP3A4
Hydrochloric Acid SCHEMBL9813887 0.99 OPRK1 (0.82) OPRK1SIGMAR1OPRM1OPRD1CYP3A4
SCHEMBL9772473 0.99 OPRK1 (0.81) OPRK1SIGMAR1OPRM1OPRD1CYP3A4
Hydrochloric Acid SCHEMBL7077496 0.99 OPRK1 (0.82) OPRK1SIGMAR1OPRM1OPRD1CYP3A4
SCHEMBL7962319 0.93 OPRK1 (0.72) OPRK1SIGMAR1OPRM1OPRD1CYP3A4
SCHEMBL9772359 0.93 OPRK1 (0.72) OPRK1SIGMAR1OPRM1OPRD1CYP3A4
SCHEMBL9748668 0.90 OPRK1 (1.00) OPRK1SIGMAR1OPRM1OPRD1CYP3A4
SCHEMBL9748062 0.90 OPRK1 (1.00) OPRK1SIGMAR1OPRM1OPRD1CYP3A4
SCHEMBL9493300 0.90 OPRK1 (0.93) OPRK1SIGMAR1OPRM1OPRD1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0258096-B1 INDANE DERIVATIVES, PROCESS FOR THEIR PREPARATION, THEIR USE AS MEDICINES, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND THE INTERMEDIATES OBTAINED ROUSSEL-UCLAF (FR) 1992-09-09 EP claimed
EP-0260555-B1 BENZO-FUSED CYCLOALKANE AND OXA- AND THIA-, CYCLOALKANE TRANS-1,2-DIAMINE DERIVATIVES THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1992-04-22 EP claimed
US-5043347-A Indanes and analgesic compositions and methods thereof ROUSSEL UCLAF (FR) 1991-08-27 US disclosed