SCHEMBL9645595

SCHEMBL9645595

CCCCCn1c(=O)[nH]c(=S)c2[nH]c(CC)nc21

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 1/20 0.42
ADORA2A P29274 1/20 0.42
PDE4B Q07343 1/20 0.42
PDE4C Q08493 1/20 0.42
PDE4D Q08499 1/20 0.42
TLR7 Q9NYK1 5/20 0.39
MAPK10 P53779 1/20 0.39
MEN1 O00255 1/20 0.39
ALDH1A1 P00352 1/20 0.39
KMT2A Q03164 1/20 0.39
HTT P42858 2/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C19 P33261 1/20 0.38
ADORA1 P30542 1/20 0.38
BRD4 O60885 1/20 0.38
BRD2 P25440 1/20 0.38
BRD3 Q15059 1/20 0.38
BRDT Q58F21 1/20 0.38
PNP P00491 1/20 0.38
TSHR P16473 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9706689 0.96 PDE4A (0.46) PDE4AADORA2APDE4BPDE4CPDE4D
SCHEMBL7420292 0.90 ADORA1 (0.44) PDE4AADORA2APDE4BPDE4CPDE4D
SCHEMBL9644450 0.86 ADORA2A (0.53) PDE4AADORA2APDE4BPDE4CPDE4D
SCHEMBL9645587 0.85 ADORA1 (0.50) ADORA2ACYP3A4CYP2C19ADORA1
SCHEMBL9706596 0.84 ADORA2A (0.41) PDE4AADORA2APDE4BPDE4CPDE4D
SCHEMBL5233098 0.84 ADORA1 (0.48) ADORA2ACYP3A4CYP2C19ADORA1
SCHEMBL9645635 0.83 ALDH1A1 (0.40) ADORA2AMEN1ALDH1A1KMT2AHTT
SCHEMBL4626790 0.82 ADORA2A (0.58) PDE4AADORA2APDE4BPDE4CPDE4D
SCHEMBL8002306 0.82 MAPT (0.39) PDE4AADORA2APDE4BPDE4CPDE4D
SCHEMBL7419694 0.81 PDE4A (0.47) PDE4AADORA2APDE4BPDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4925847-A BRONCHODILATORS EUROCELTIQUE, S.A. (LU) 1990-05-15 US claimed
EP-0256692-B1 6-THIOXANTHINES Euroceltique S.A. (LU) 1992-09-16 EP disclosed
US-5010081-A Bronchodilator agents EUROCELTIQUE, S.A. (LU) 1991-04-23 US disclosed
US-4925847-A BRONCHODILATORS EUROCELTIQUE, S.A. (LU) 1990-05-15 US disclosed
EP-0256692-A2 6-Thioxanthines Euroceltique S.A. (LU) 1988-02-24 EP disclosed