SCHEMBL9651995

SCHEMBL9651995

NC(=O)N1CCN(C(=O)Cc2ccc(Cl)c(Cl)c2)C(CN2CCCC2)C1

nearest known ligand 0.81

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRK1 P41145 17/20 0.81
OPRM1 P35372 2/20 0.76
CYP3A4 P08684 2/20 0.76
CYP2D6 P10635 2/20 0.76
CYP2C9 P11712 2/20 0.76
CYP2C19 P33261 2/20 0.76
OPRD1 P41143 2/20 0.76
TDP1 Q9NUW8 2/20 0.76
NPC1 O15118 1/20 0.69
CYP1A2 P05177 1/20 0.69
NFKB1 P19838 1/20 0.69
HIF1A Q16665 1/20 0.69
BLM P54132 2/20 0.69
MEN1 O00255 1/20 0.69
LMNA P02545 1/20 0.69
MAPK1 P28482 1/20 0.69
KMT2A Q03164 1/20 0.69
NPSR1 Q6W5P4 1/20 0.69
PMP22 Q01453 1/20 0.68
DRD4 P21917 1/20 0.68

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6359486 0.99 OPRK1 (0.79) OPRK1OPRM1CYP3A4CYP2D6CYP2C9
Hydrochloric Acid SCHEMBL5629280 0.99 OPRK1 (0.79) OPRK1OPRM1CYP3A4CYP2D6CYP2C9
SCHEMBL2683751 0.90 OPRK1 (0.82) OPRK1OPRM1CYP3A4CYP2D6CYP2C9
SCHEMBL8221866 0.89 OPRK1 (1.00) OPRK1OPRM1CYP3A4CYP2D6CYP2C9
SCHEMBL8221863 0.89 OPRK1 (1.00) OPRK1OPRM1CYP3A4CYP2D6CYP2C9
SCHEMBL10417791 0.88 OPRK1 (1.00) OPRK1OPRM1CYP3A4CYP2D6CYP2C9
Hydrochloric Acid SCHEMBL5629721 0.88 OPRK1 (0.98) OPRK1OPRM1CYP3A4CYP2D6CYP2C9
Hydrochloric Acid SCHEMBL5629714 0.88 OPRK1 (0.98) OPRK1OPRM1CYP3A4CYP2D6CYP2C9
SCHEMBL10416654 0.88 OPRK1 (1.00) OPRK1OPRM1CYP3A4CYP2D6CYP2C9
SCHEMBL4545382 0.87 OPRK1 (1.00) OPRK1OPRM1CYP3A4CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5116842-A Analgesics GLAXO GROUP LIMITED (GB) 1992-05-26 US disclosed
EP-0398720-A2 Piperazine derivatives GLAXO GROUP LIMITED (GB) 1990-11-22 EP disclosed