SCHEMBL9657352

SCHEMBL9657352

O=C1c2ccccc2C(=O)N1Nc1ccc(O)cc1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.71
RPS6KA2 Q15349 1/20 0.57
ALDH1A1 P00352 4/20 0.54
MAPT P10636 8/20 0.49
POLB P06746 2/20 0.48
CASP6 P55212 1/20 0.47
MAPK1 P28482 3/20 0.45
RAB9A P51151 3/20 0.45
NPSR1 Q6W5P4 2/20 0.45
NR1H3 Q13133 1/20 0.45
PTGS1 P23219 1/20 0.45
PTGS2 P35354 1/20 0.45
NPC1 O15118 1/20 0.45
GAA P10253 1/20 0.45
HTT P42858 1/20 0.45
MEN1 O00255 4/20 0.44
KMT2A Q03164 4/20 0.44
KDM4E B2RXH2 3/20 0.44
TDP1 Q9NUW8 2/20 0.44
JAK2 O60674 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3259551 0.84 CYP1A2 (1.00) CYP1A2ALDH1A1MAPTCASP6RAB9A
SCHEMBL14322059 0.82 CYP1A2 (0.74) CYP1A2ALDH1A1MAPTCASP6NPSR1
Hydrochloric Acid SCHEMBL5138493 0.82 CYP1A2 (0.96) CYP1A2ALDH1A1MAPTCASP6RAB9A
SCHEMBL133402 0.81 CYP1A2 (0.71) CYP1A2RPS6KA2ALDH1A1MAPTPOLB
SCHEMBL20945035 0.80 CYP1A2 (0.70) CYP1A2ALDH1A1MAPTPOLBCASP6
SCHEMBL7485009 0.77 CYP1A2 (0.71) CYP1A2ALDH1A1MAPTCASP6RAB9A
SCHEMBL21026687 0.77 CYP1A2 (0.70) CYP1A2RPS6KA2ALDH1A1MAPTCASP6
SCHEMBL5821136 0.77 CYP1A2 (0.65) CYP1A2RPS6KA2ALDH1A1MAPTPOLB
SCHEMBL14321431 0.77 CYP1A2 (0.65) CYP1A2RPS6KA2ALDH1A1MAPTCASP6
SCHEMBL20945151 0.76 MAPK1 (0.59) CYP1A2ALDH1A1MAPTPOLBMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0516588-A1 Substituted diaminophtalimides and analogues CIBA-GEIGY AG (CH) 1992-12-02 EP disclosed