SCHEMBL5821136

SCHEMBL5821136

COc1ccc(NN2C(=O)c3ccccc3C2=O)cc1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.65
RPS6KA2 Q15349 2/20 0.60
MAPT P10636 4/20 0.55
ALDH1A1 P00352 3/20 0.51
RAB9A P51151 2/20 0.51
MAPK1 P28482 2/20 0.51
KDM4E B2RXH2 1/20 0.51
NSD2 O96028 1/20 0.51
LMNA P02545 1/20 0.51
POLB P06746 1/20 0.51
HPGD P15428 1/20 0.51
HTT P42858 1/20 0.51
SMN1; SMN2 Q16637 1/20 0.51
TDP1 Q9NUW8 1/20 0.51
L3MBTL1 Q9Y468 1/20 0.51
NR1H3 Q13133 2/20 0.49
APP P05067 1/20 0.49
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
CASP3 P42574 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21026687 0.83 CYP1A2 (0.70) CYP1A2RPS6KA2MAPTALDH1A1HPGD
SCHEMBL3259551 0.79 CYP1A2 (1.00) CYP1A2MAPTALDH1A1RAB9AKDM4E
SCHEMBL20945151 0.79 MAPK1 (0.59) CYP1A2MAPTALDH1A1MAPK1KDM4E
SCHEMBL14322059 0.78 CYP1A2 (0.74) CYP1A2MAPTALDH1A1KDM4ELMNA
Hydrochloric Acid SCHEMBL5138493 0.77 CYP1A2 (0.96) CYP1A2MAPTALDH1A1RAB9AKDM4E
SCHEMBL11403753 0.77 CYP1A2 (0.59) CYP1A2RPS6KA2MAPTALDH1A1RAB9A
SCHEMBL9657352 0.77 CYP1A2 (0.71) CYP1A2RPS6KA2MAPTALDH1A1RAB9A
SCHEMBL133402 0.77 CYP1A2 (0.71) CYP1A2RPS6KA2MAPTALDH1A1RAB9A
SCHEMBL28085321 0.77 MGLL (0.53) RPS6KA2MAPTALDH1A1RAB9AMAPK1
SCHEMBL9656206 0.76 CYP1A2 (0.60) CYP1A2ALDH1A1RAB9AHPGDSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006047514-A2 DAPH ANALOGS AND INHIBITION OF PROTEIN AGGREGATION WHITEHEAD INSTITUTE FOR BIOMEDICAL RESEARCH (US) 2006-05-04 WO disclosed