SCHEMBL9664101

SCHEMBL9664101

C=C1N(C)C(=O)CC12CCN(Cc1ccccc1)CC2

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 11/20 0.49
DRD2 P14416 3/20 0.49
HTR2A P28223 3/20 0.49
HTR2C P28335 3/20 0.49
HTR2B P41595 3/20 0.49
CYP3A4 P08684 4/20 0.47
CYP2D6 P10635 4/20 0.47
CYP2C19 P33261 4/20 0.47
TSHR P16473 3/20 0.47
CYP2C9 P11712 3/20 0.47
TP53 P04637 2/20 0.47
CYP1A2 P05177 2/20 0.47
ALDH1A1 P00352 2/20 0.47
HSD17B10 Q99714 1/20 0.47
MC4R P32245 1/20 0.46
OPRL1 P41146 2/20 0.45
OPRM1 P35372 1/20 0.45
OPRD1 P41143 1/20 0.45
OPRK1 P41145 1/20 0.45
NFKB1 P19838 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6777379 0.78 SIGMAR1 (0.60) SIGMAR1DRD2HTR2AHTR2CHTR2B
SCHEMBL12846708 0.76 CHRM2 (0.58) SIGMAR1DRD2HTR2AHTR2CHTR2B
SCHEMBL7290398 0.75 SIGMAR1 (0.55) SIGMAR1DRD2CYP3A4HSD17B10
Hydrochloric Acid SCHEMBL10566456 0.74 SIGMAR1 (0.49) SIGMAR1DRD2HTR2AHTR2CHTR2B
SCHEMBL24994297 0.72 CYP2D6 (0.55) SIGMAR1CYP3A4CYP2D6CYP2C19TSHR
SCHEMBL1042820 0.71 SIGMAR1 (0.53) SIGMAR1DRD2HTR2AHTR2CHTR2B
SCHEMBL10567177 0.71 SIGMAR1 (0.47) SIGMAR1DRD2HTR2AHTR2CHTR2B
SCHEMBL28978295 0.71 MEN1 (0.58) SIGMAR1DRD2HTR2AHTR2CHTR2B
SCHEMBL1223370 0.70 SIGMAR1 (0.52) SIGMAR1DRD2HTR2AHTR2CHTR2B
SCHEMBL1344124 0.70 SIGMAR1 (0.55) SIGMAR1DRD2HTR2AHTR2CHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5157038-A Antidepressants; tranquilizers; treatment of schizophrenia and epilepsy; antilepmic agents RICHTER GEDEON VEGYESZETI GYAR RT. (HU) 1992-10-20 US disclosed