SCHEMBL9664994

SCHEMBL9664994

Cc1nc2ccc(Cn3ccnc3)cc2n1O

nearest known ligand 0.52

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 9/20 0.52
CYP11B1 P15538 9/20 0.52
CYP11B2 P19099 9/20 0.52
TBXAS1 P24557 2/20 0.49
ADRA2C P18825 1/20 0.48
CYP2A6 P11509 1/20 0.47
CYP2B6 P20813 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9662260 0.88 CYP19A1 (0.51) CYP19A1CYP11B1CYP11B2TBXAS1ADRA2C
SCHEMBL9664756 0.85 CYP19A1 (0.54) CYP19A1CYP11B1CYP11B2TBXAS1ADRA2C
SCHEMBL9664806 0.84 KCNH2 (0.50) CYP19A1CYP11B1CYP11B2TBXAS1CYP2A6
SCHEMBL9664986 0.83 CYP11B1 (0.56) CYP19A1CYP11B1CYP11B2TBXAS1
Water SCHEMBL9664102 0.82 CYP11B1 (0.54) CYP19A1CYP11B1CYP11B2TBXAS1
SCHEMBL9663632 0.81 CYP11B1 (0.56) CYP19A1CYP11B1CYP11B2TBXAS1
SCHEMBL9662930 0.80 CYP19A1 (0.54) CYP19A1CYP11B1CYP11B2TBXAS1ADRA2C
SCHEMBL9663739 0.80 CYP11B1 (0.53) CYP19A1CYP11B1CYP11B2TBXAS1
SCHEMBL9662907 0.77 CCNT1 (0.46) CYP19A1CYP11B1CYP11B2TBXAS1ADRA2C
SCHEMBL9665025 0.76 CYP19A1 (0.45) CYP19A1CYP11B1CYP11B2TBXAS1ADRA2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0260744-B1 (1H-IMIDAZOL-1-YLMETHYL) SUBSTITUTED BENZIMIDAZOLE DERIVATIVES JANSSEN PHARMACEUTICA N.V. (BE) 1992-12-16 EP disclosed
US-4859684-A (1H-imidazol-1-ylmethyl) substituted benzimidazole derivatives and use thereof in treating androgen dependent disorders JANSSEN PHARMACEUTICA N.V. (BE) 1989-08-22 US disclosed
EP-0260744-A2 (1H-imidazol-1-ylmethyl) substituted benzimidazole derivatives JANSSEN PHARMACEUTICA N.V. (BE) 1988-03-23 EP disclosed