SCHEMBL9668673

SCHEMBL9668673

Clc1cnc(-c2ncc[nH]2)[nH]1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 2/20 0.55
PDE4B Q07343 2/20 0.55
PDE4C Q08493 2/20 0.55
PDE4D Q08499 2/20 0.55
NISCH Q9Y2I1 2/20 0.41
MTOR P42345 1/20 0.41
ADK P55263 1/20 0.41
ALDH1A1 P00352 4/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
IDO1 P14902 1/20 0.35
KDM4E B2RXH2 2/20 0.34
CHEK1 O14757 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.33
SMPD3 Q9NY59 1/20 0.33
ADRA2A P08913 2/20 0.32
CSNK1A1 P48729 1/20 0.32
TYRO3 Q06418 1/20 0.32
DYRK1B Q9Y463 1/20 0.32
CYP1A2 P05177 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL81650 0.76 NISCH (0.59) PDE4APDE4BPDE4CPDE4DNISCH
SCHEMBL28425230 0.74 NISCH (0.56) PDE4APDE4BPDE4CPDE4DNISCH
Hydrochloric Acid SCHEMBL1536214 0.74 NISCH (0.56) PDE4APDE4BPDE4CPDE4DNISCH
SCHEMBL5454911 0.71 NISCH (0.45) PDE4APDE4BPDE4CPDE4DNISCH
SCHEMBL10720400 0.71 PDE4A (1.00) PDE4APDE4BPDE4CPDE4DNISCH
SCHEMBL10768507 0.68 PDE4A (0.47) PDE4APDE4BPDE4CPDE4DNISCH
SCHEMBL20595279 0.67 PDE4A (0.46) PDE4APDE4BPDE4CPDE4DNISCH
SCHEMBL20595281 0.67 PDE4A (0.46) PDE4APDE4BPDE4CPDE4DNISCH
SCHEMBL28536155 0.64 NPY5R (0.59) MTORKMT2AKDM4ESMN1; SMN2CYP1A2
SCHEMBL29432814 0.64 NISCH (0.42) PDE4APDE4BPDE4CPDE4DNISCH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0229922-B1 NOVEL 2,2'-BI-1H-IMIDAZOLES MERRELL DOW PHARMACEUTICALS INC. (US) 1992-04-15 EP disclosed
EP-0229922-A2 Novel 2,2'-BI-1H-imidazoles MERRELL DOW PHARMACEUTICALS INC. (US) 1987-07-29 EP disclosed