SCHEMBL9669264

SCHEMBL9669264

O=Cc1cc([N+](=O)[O-])cc2ccccc12

nearest known ligand 0.62

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 2/20 0.62
TSHR P16473 1/20 0.62
CYP3A4 P08684 1/20 0.50
ERN1 O75460 3/20 0.49
KMT2A Q03164 5/20 0.45
MEN1 O00255 4/20 0.45
PTPN1 P18031 1/20 0.45
ALDH1A1 P00352 6/20 0.45
SMN1; SMN2 Q16637 3/20 0.45
LMNA P02545 3/20 0.45
MAPT P10636 2/20 0.45
KDM4E B2RXH2 1/20 0.45
HTT P42858 1/20 0.45
ALOX5 P09917 3/20 0.44
PTGES O14684 1/20 0.44
RXRA P19793 1/20 0.44
CASP6 P55212 1/20 0.44
RAB9A P51151 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4872775 0.81 ERN1 (0.51) TDP1TSHRCYP3A4ERN1KMT2A
SCHEMBL17348536 0.81 TDP1 (0.55) TDP1TSHRCYP3A4KMT2AMEN1
Dinitrophenylene SCHEMBL27328531 0.80 ALDH1A1 (0.59) TDP1TSHRCYP3A4ERN1KMT2A
SCHEMBL5248911 0.79 TSHR (0.66) TDP1TSHRCYP3A4KMT2AMEN1
SCHEMBL17348528 0.78 ERN1 (0.44) TDP1TSHRERN1PTPN1ALDH1A1
SCHEMBL57381 0.77 TDP1 (1.00) TDP1TSHRCYP3A4KMT2AMEN1
SCHEMBL29475186 0.77 TDP1 (1.00) TDP1TSHRCYP3A4KMT2AMEN1
SCHEMBL1378334 0.75 TDP1 (0.66) TDP1TSHRCYP3A4KMT2AMEN1
SCHEMBL17599539 0.75 TSHR (0.66) TDP1TSHRCYP3A4KMT2AMEN1
SCHEMBL4960980 0.75 TDP1 (0.66) TDP1TSHRCYP3A4KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104072493-B Naphthalimide compound containing 2-mercaptobenzothiazole and triazole heterocycle, preparation method and application thereof 大连理工大学 2017-01-04 CN disclosed
WO-2015191640-A2 BICYCLIC XANTHINE OXIDASE INHIBITORS AND METHODS OF USE BAYLOR COLLEGE OF MEDICINE (US) 2015-12-17 WO disclosed
US-5155113-A Administering 5-fluorouracil and derivatives with pyridine and pyridone derivatives OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1992-10-13 US disclosed
EP-0180188-B1 A COMPOSITION FOR INCREASING THE ANTI-CANCER ACTIVITY OF AN ANTI-CANCER COMPOUND OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1992-04-15 EP disclosed
EP-0180188-A2 A composition for increasing the anti-cancer activity of an anti-cancer compound OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1986-05-07 EP disclosed