SCHEMBL9669372

SCHEMBL9669372

Cc1nnc2n1-c1sc(CCCO)cc1C(c1ccccc1Cl)=NC2

nearest known ligand 0.76

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
OPRK1 P41145 1/20 0.76
PDE4D Q08499 1/20 0.76
PTAFR P25105 19/20 0.74
CYP3A4 P08684 1/20 0.68
ALOX15 P16050 1/20 0.68

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10471373 0.97 OPRK1 (0.75) OPRK1PDE4DPTAFRCYP3A4ALOX15
SCHEMBL9667874 0.96 OPRK1 (0.74) OPRK1PDE4DPTAFRCYP3A4ALOX15
SCHEMBL10471499 0.96 OPRK1 (0.74) OPRK1PDE4DPTAFRCYP3A4ALOX15
SCHEMBL10469753 0.96 OPRK1 (0.74) OPRK1PDE4DPTAFRCYP3A4ALOX15
SCHEMBL10469718 0.91 PTAFR (0.88) OPRK1PDE4DPTAFRCYP3A4ALOX15
SCHEMBL10471094 0.90 OPRK1 (0.76) OPRK1PDE4DPTAFRCYP3A4ALOX15
SCHEMBL9525884 0.89 PTAFR (0.81) OPRK1PDE4DPTAFRCYP3A4ALOX15
SCHEMBL10464347 0.89 PTAFR (0.81) OPRK1PDE4DPTAFRCYP3A4ALOX15
SCHEMBL9525077 0.89 PTAFR (0.81) OPRK1PDE4DPTAFRCYP3A4ALOX15
SCHEMBL9522397 0.89 PTAFR (0.81) OPRK1PDE4DPTAFRCYP3A4ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0230942-B1 THIENO-1,4-DIAZEPINES BOEHRINGER INGELHEIM KG (DE) 1992-04-29 EP disclosed
US-4900729-A PLATELET ACTIVATING FACTOR ANTAGONISTS BOEHRINGER INGELHEIM KG (DE) 1990-02-13 US disclosed
EP-0230942-A2 Thieno-1,4-diazepines BOEHRINGER INGELHEIM KG (DE) 1987-08-05 EP disclosed