SCHEMBL9675562

SCHEMBL9675562

Cc1c(F)c(N)cc([N+](=O)[O-])c1F

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TSHR P16473 5/20 0.48
CYP3A4 P08684 5/20 0.44
ALDH1A1 P00352 4/20 0.44
RECQL P46063 1/20 0.44
TDP1 Q9NUW8 7/20 0.42
MEN1 O00255 1/20 0.42
POLB P06746 1/20 0.42
MAPT P10636 1/20 0.42
KMT2A Q03164 1/20 0.42
ALOX15 P16050 1/20 0.42
CYP1A2 P05177 2/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
GPR35 Q9HC97 2/20 0.39
ATM Q13315 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30237358 0.86 TSHR (0.47) TSHRCYP3A4ALDH1A1RECQLTDP1
SCHEMBL9676449 0.85 TDP1 (0.50) TSHRCYP3A4ALDH1A1RECQLTDP1
SCHEMBL19501351 0.80 TSHR (0.48) TSHRCYP3A4ALDH1A1RECQLTDP1
SCHEMBL1505782 0.79 TDP1 (0.45) TSHRCYP3A4ALDH1A1RECQLTDP1
SCHEMBL27768818 0.78 TSHR (0.47) TSHRCYP3A4ALDH1A1RECQLTDP1
SCHEMBL21373613 0.78 TSHR (0.52) TSHRCYP3A4ALDH1A1RECQLTDP1
SCHEMBL28102481 0.78 ALDH1A1 (0.44) TSHRCYP3A4ALDH1A1TDP1MEN1
SCHEMBL31543948 0.78 CYP1A2 (0.47) TSHRCYP3A4ALDH1A1RECQLTDP1
SCHEMBL30857795 0.76 TSHR (0.53) TSHRCYP3A4ALDH1A1RECQLTDP1
SCHEMBL1635417 0.76 TSHR (0.53) TSHRCYP3A4ALDH1A1RECQLTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0237955-B1 QUINOLONECARBOXYLIC ACID DERIVATIVES AND THEIR PREPARATION KYORIN PHARMACEUTICAL CO., LTD. (JP) 1992-07-15 EP disclosed
US-4894458-A BACTERICIDES KYORIN PHARMACEUTICAL CO., LTD. (JP) 1990-01-16 US disclosed
EP-0237955-A2 Quinolonecarboxylic acid derivatives and their preparation KYORIN PHARMACEUTICAL CO., LTD. (JP) 1987-09-23 EP disclosed