SCHEMBL9680326

SCHEMBL9680326

CC(=O)c1cc(N)c(=O)[nH]c1C

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 4/20 0.57
GAA P10253 5/20 0.50
NPC1 O15118 1/20 0.50
POLB P06746 1/20 0.50
PDE3B Q13370 2/20 0.46
PDE3A Q14432 2/20 0.46
PDE4A P27815 1/20 0.46
PDE4B Q07343 1/20 0.46
PDE4C Q08493 1/20 0.46
PDE4D Q08499 1/20 0.46
AURKB Q96GD4 1/20 0.44
INCENP Q9NQS7 1/20 0.44
KDM4E B2RXH2 3/20 0.43
HSD17B10 Q99714 3/20 0.43
HPGD P15428 2/20 0.43
ALDH1A1 P00352 2/20 0.42
MAPT P10636 2/20 0.42
LMNA P02545 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9476064 0.98 BRD4 (0.55) BRD4GAANPC1POLBPDE3B
SCHEMBL9477063 0.80 GAA (0.55) BRD4GAANPC1POLBPDE3B
SCHEMBL9475536 0.79 GAA (0.57) BRD4GAANPC1POLBKDM4E
SCHEMBL9475977 0.77 KDM4E (0.67) BRD4GAANPC1POLBKDM4E
SCHEMBL10675219 0.76 MAPT (0.54) BRD4GAAPOLBPDE3BPDE3A
SCHEMBL4514368 0.73 KDM4E (0.50) GAANPC1POLBPDE3BPDE3A
SCHEMBL18044655 0.73 GAA (0.62) BRD4GAANPC1POLBPDE3B
SCHEMBL9846132 0.73 PDE3B (0.53) GAAPDE3BPDE3APDE4APDE4B
SCHEMBL3678604 0.73 BRD4 (0.47) BRD4GAANPC1POLBKDM4E
SCHEMBL13995853 0.72 GAA (0.71) BRD4GAANPC1POLBKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4568751-A 5-Acyl-2-(1H)-pyridinones MERRELL DOW PHARMACEUTICALS INC. (US) 1986-02-04 US claimed
EP-0481802-A1 Hydroxylated inhibitors of HIV reverse transcriptase MERCK & CO. INC. (US) 1992-04-22 EP disclosed