SCHEMBL9680408

SCHEMBL9680408

O=C(O)C1CCC(COc2ccc(Cl)cc2)CC1

nearest known ligand 0.56

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PARP15 Q460N3 4/20 0.54
PARP10 Q53GL7 4/20 0.54
PARP2 Q9UGN5 2/20 0.54
CYP4F2 P78329 1/20 0.52
CYP4A11 Q02928 1/20 0.52
ATF4 P18848 3/20 0.50
S1PR5 Q9H228 1/20 0.47
FFAR4 Q5NUL3 1/20 0.46
LTA4H P09960 2/20 0.45
MAPT P10636 1/20 0.44
CXCR3 P49682 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3667235 0.85 PARP15 (0.55) PARP15PARP10PARP2ATF4LTA4H
SCHEMBL10207302 0.82 PARP15 (0.51) PARP15PARP10PARP2CYP4F2CYP4A11
SCHEMBL765066 0.82 PARP15 (0.51) PARP15PARP10PARP2CYP4F2CYP4A11
SCHEMBL10203545 0.79 ACACB (0.59) PARP15PARP10PARP2CYP4F2CYP4A11
SCHEMBL879115 0.79 ACACB (0.59) PARP15PARP10PARP2CYP4F2CYP4A11
SCHEMBL4186691 0.76 PARP15 (0.58) PARP15PARP10PARP2LTA4H
SCHEMBL29082785 0.76 ATF4 (0.84) ATF4
SCHEMBL21413242 0.76 CYP4F2 (0.47) PARP15PARP10PARP2CYP4F2CYP4A11
SCHEMBL29024848 0.75 PARP15 (0.64) PARP15PARP10PARP2
SCHEMBL416244 0.75 PARP15 (0.72) PARP15PARP10PARP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5175319-A Antiprotozoa agent, useful for treating malaria, theileriosis, coccidiosis and prophylaxix BURROUGHS WELLCOME CO. (US) 1992-12-29 US disclosed
US-5053432-A Antiprotozoa agents; treatment of malaria BURROUGHS WELLCOME CO. (US) 1991-10-01 US disclosed
EP-0123238-B1 NAPHTHOQUINONE DERIVATIVES THE WELLCOME FOUNDATION LIMITED (GB) 1987-06-10 EP disclosed
EP-0123238-A2 Naphthoquinone derivatives THE WELLCOME FOUNDATION LIMITED (GB) 1984-10-31 EP disclosed