SCHEMBL9680862

SCHEMBL9680862

CN=C=O.c1cc2ccc1-2

nearest known ligand 0.60

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.60
CASP1 P29466 1/20 0.60
CYP3A4 P08684 4/20 0.37
ALDH1A1 P00352 2/20 0.37
TDP1 Q9NUW8 2/20 0.37
HPGD P15428 1/20 0.37
HRH3 Q9Y5N1 3/20 0.33
GABRA1 P14867 1/20 0.32
GABRB2 P47870 1/20 0.32
HTT P42858 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
TP53 P04637 1/20 0.30
ESR1 P03372 1/20 0.30
ESR2 Q92731 1/20 0.30
TRPA1 O75762 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9743213 0.91 TSHR (0.50) TSHRCASP1CYP3A4ALDH1A1TDP1
Biphenyl SCHEMBL1840808 0.85 ALDH1A1 (0.50) TSHRCASP1CYP3A4ALDH1A1TDP1
SCHEMBL27363200 0.78 TSHR (0.82) TSHRCASP1ALDH1A1
SCHEMBL2765 0.78
SCHEMBL28124906 0.78
SCHEMBL9679096 0.77 TSHR (0.47) TSHRCASP1CYP3A4ALDH1A1TDP1
Ethane SCHEMBL6257492 0.76 SMN1; SMN2 (0.32) CYP3A4ALDH1A1TDP1HTTSMN1; SMN2
Benzene SCHEMBL27960086 0.74 TSHR (0.75) TSHRCASP1CYP3A4ALDH1A1GABRA1
Benzene SCHEMBL9680470 0.74 TSHR (0.75) TSHRCASP1CYP3A4ALDH1A1GABRA1
SCHEMBL1502365 0.73

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5082937-A Gastrin or cholecystokinin antagonists JOUVEINAL S.A. (FR) 1992-01-21 US disclosed
EP-0420716-A2 Benzodiazepines, process and intermediates for their preparation and their therapeutic use JOUVEINAL S.A. (FR) 1991-04-03 EP disclosed