SCHEMBL9681055

SCHEMBL9681055

Nc1cccc(C#Cc2ccc(F)c([N+](=O)[O-])c2)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.46
HIF1A Q16665 1/20 0.46
VCAM1 P19320 1/20 0.44
FFAR1 O14842 1/20 0.42
TDP1 Q9NUW8 3/20 0.40
CYP3A4 P08684 2/20 0.40
ALOX15 P16050 2/20 0.40
TSHR P16473 2/20 0.40
L3MBTL1 Q9Y468 2/20 0.40
PDE7A Q13946 1/20 0.40
ADRB2 P07550 1/20 0.40
RAB9A P51151 1/20 0.40
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA9 Q16790 1/20 0.39
MAPT P10636 3/20 0.39
LMNA P02545 2/20 0.39
HTT P42858 2/20 0.39
MEN1 O00255 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2426169 0.86 ALDH1A1 (0.60) ALDH1A1HIF1AVCAM1TDP1CA1
SCHEMBL9679775 0.77 FFAR1 (0.46) ALDH1A1FFAR1CYP3A4L3MBTL1ADRB2
SCHEMBL394329 0.77 ALDH1A1 (0.64) ALDH1A1HIF1AVCAM1TDP1CYP3A4
SCHEMBL4408381 0.77 TDP1 (0.51) ALDH1A1HIF1AVCAM1TDP1CYP3A4
SCHEMBL13622489 0.76 ALDH1A1 (0.70) ALDH1A1FFAR1TDP1ALOX15TSHR
SCHEMBL4971914 0.76 PIK3CA (0.45) ALDH1A1FFAR1CYP3A4L3MBTL1ADRB2
SCHEMBL1027029 0.75 ALDH1A1 (0.37) ALDH1A1FFAR1TDP1CYP3A4ALOX15
SCHEMBL697848 0.74 ALDH1A1 (0.58) ALDH1A1HIF1AVCAM1TDP1CA1
SCHEMBL9611202 0.73 FFAR1 (0.59) ALDH1A1FFAR1TDP1CYP3A4L3MBTL1
SCHEMBL4968126 0.73 CYP3A4 (0.58) ALDH1A1FFAR1TDP1CYP3A4L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0493650-A1 Fluorinated acetylene-containing aromatic amines and diamines National Starch and Chemical Investment Holding Corporation (US) 1992-07-08 EP claimed
US-5107026-A Fluorinated acetylene-containing aromatic amines and diamines NATIONAL STARCH AND CHEMICAL INVESTMENT HOLDING CORPORATION (US) 1992-04-21 US claimed
EP-0493650-A1 Fluorinated acetylene-containing aromatic amines and diamines National Starch and Chemical Investment Holding Corporation (US) 1992-07-08 EP disclosed
US-5107026-A Fluorinated acetylene-containing aromatic amines and diamines NATIONAL STARCH AND CHEMICAL INVESTMENT HOLDING CORPORATION (US) 1992-04-21 US disclosed