SCHEMBL9681219

SCHEMBL9681219

COc1ccc(-n2nc(N3CCNCC3)c3ccccc32)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KHK P50053 7/20 0.56
ADRB1 P08588 3/20 0.55
HTR3A P46098 2/20 0.55
HTR3E A5X5Y0 1/20 0.55
HTR3B O95264 1/20 0.55
HTR3D Q70Z44 1/20 0.55
HTR3C Q8WXA8 1/20 0.55
SIGMAR1 Q99720 1/20 0.55
HTR1A P08908 3/20 0.46
HTR7 P34969 2/20 0.46
CYP1A2 P05177 2/20 0.45
CYP3A4 P08684 2/20 0.45
CYP2D6 P10635 2/20 0.45
TSHR P16473 2/20 0.45
TP53 P04637 1/20 0.45
SLC2A1 P11166 1/20 0.45
SLC2A2 P11168 1/20 0.45
SLC2A3 P11169 1/20 0.45
MEN1 O00255 1/20 0.44
USP2 O75604 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9681291 0.99 KHK (0.55) KHKADRB1HTR3AHTR3EHTR3B
SCHEMBL9681274 0.86 HRH4 (0.49) KHKCYP1A2CYP3A4CYP2D6TSHR
SCHEMBL9681867 0.86 KHK (0.53) KHKADRB1HTR3A
SCHEMBL2710715 0.85 KHK (0.54) KHKADRB1HTR3AHTR3EHTR3B
Hydrochloric Acid SCHEMBL9680640 0.85 HRH4 (0.48) KHKCYP1A2CYP3A4CYP2D6TSHR
Hydrochloric Acid SCHEMBL9680719 0.85 KHK (0.52) KHKADRB1HTR3AHTR1ACYP1A2
Hydrochloric Acid SCHEMBL9681346 0.84 KHK (0.53) KHKADRB1HTR3AHTR3EHTR3B
SCHEMBL9681720 0.83 KHK (0.47) KHKADRB1HTR3AHTR3EHTR3B
SCHEMBL9681305 0.83 KHK (0.47) KHKHTR3AHTR1AHTR7HTR6
SCHEMBL9681327 0.83 KHK (0.47) KHKHTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4999356-A Analgesics, antidepressants, anticonvulsants HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1991-03-12 US claimed
US-5134236-A Analgesics, antidepressants, anticonvulsants HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1992-07-28 US disclosed
US-4999356-A Analgesics, antidepressants, anticonvulsants HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1991-03-12 US disclosed
EP-0302423-A2 1-Phenyl-3-(1-piperazinyl)-1h-indazoles, a process and intermediates for their preparation, and the use thereof as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1989-02-08 EP disclosed