SCHEMBL9681305

SCHEMBL9681305

Fc1ccc(-n2nc(N3CCNCC3)c3ccccc32)cc1

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KHK P50053 7/20 0.47
HTR3A P46098 1/20 0.45
HTR6 P50406 1/20 0.44
HTR7 P34969 2/20 0.43
HTR2C P28335 1/20 0.43
HRH4 Q9H3N8 1/20 0.42
HRH3 Q9Y5N1 1/20 0.42
HTR1A P08908 2/20 0.42
KDM4E B2RXH2 1/20 0.42
MAPT P10636 1/20 0.42
SLC6A2 P23975 1/20 0.41
SLC6A4 P31645 1/20 0.41
SLC6A3 Q01959 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2710715 0.89 KHK (0.54) KHKHTR3AHTR6HTR2CKDM4E
Hydrochloric Acid SCHEMBL9681346 0.87 KHK (0.53) KHKHTR3AHTR6HTR2CKDM4E
SCHEMBL9681327 0.86 KHK (0.47) KHKHTR6HTR2CHRH4KDM4E
SCHEMBL9683240 0.86 KHK (0.50) KHKHTR6HTR7HRH4HRH3
SCHEMBL9681867 0.86 KHK (0.53) KHKHTR3AHTR2C
SCHEMBL9681720 0.86 KHK (0.47) KHKHTR3AHTR6HTR2CKDM4E
SCHEMBL9682489 0.86 HTR6 (0.47) KHKHTR3AHTR6HTR2CHRH4
SCHEMBL9682462 0.86 KHK (0.44) KHKHTR3AHTR6HTR7HTR2C
Hydrochloric Acid SCHEMBL9680719 0.85 KHK (0.52) KHKHTR3AHTR2CHTR1AKDM4E
Hydrochloric Acid SCHEMBL9680573 0.85 HTR6 (0.46) KHKHTR3AHTR6HTR2CHRH4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4999356-A Analgesics, antidepressants, anticonvulsants HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1991-03-12 US claimed
US-5134236-A Analgesics, antidepressants, anticonvulsants HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1992-07-28 US disclosed
US-4999356-A Analgesics, antidepressants, anticonvulsants HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1991-03-12 US disclosed
EP-0302423-A2 1-Phenyl-3-(1-piperazinyl)-1h-indazoles, a process and intermediates for their preparation, and the use thereof as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1989-02-08 EP disclosed