SCHEMBL9682518

SCHEMBL9682518

CCOC(=O)N1CCN(c2nn(-c3ccc(C(F)(F)F)cc3)c3ccccc23)CC1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 4/20 0.53
HPGD P15428 4/20 0.53
KMT2A Q03164 7/20 0.50
MEN1 O00255 6/20 0.50
ALDH1A1 P00352 4/20 0.48
POLB P06746 2/20 0.48
ADRB2 P07550 1/20 0.48
TSHR P16473 2/20 0.47
HSD17B10 Q99714 2/20 0.47
ALOX15 P16050 1/20 0.47
RXFP1 Q9HBX9 1/20 0.47
PDK2 Q15119 1/20 0.46
MAPT P10636 4/20 0.45
LMNA P02545 2/20 0.45
HTT P42858 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
GAA P10253 2/20 0.45
KDM4E B2RXH2 1/20 0.45
TACR1 P25103 1/20 0.44
MAPK1 P28482 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9682148 0.89 KMT2A (0.52) SMN1; SMN2HPGDKMT2AMEN1ALDH1A1
SCHEMBL9681416 0.88 KMT2A (0.58) SMN1; SMN2HPGDKMT2AMEN1ALDH1A1
SCHEMBL9763297 0.84 SCN9A (0.46) SMN1; SMN2KMT2AMAPTLMNANPSR1
SCHEMBL9763384 0.82 KHK (0.48) SMN1; SMN2KMT2AMEN1ALDH1A1MAPT
SCHEMBL9680624 0.81 CYP1A2 (0.46) KMT2AMEN1ADRB2TSHRHSD17B10
Fumaric Acid SCHEMBL9681243 0.80 KHK (0.44) KMT2AMEN1ALDH1A1ADRB2LMNA
Fumaric Acid SCHEMBL9681235 0.80 KHK (0.44) KMT2AMEN1ALDH1A1ADRB2LMNA
SCHEMBL30627066 0.79 MAPT (0.69) SMN1; SMN2HPGDKMT2AMEN1ALDH1A1
Fumaric Acid SCHEMBL9680682 0.79 KDM4E (0.54) KMT2AMEN1ALDH1A1ADRB2TSHR
Fumaric Acid SCHEMBL9680687 0.79 KDM4E (0.54) KMT2AMEN1ALDH1A1ADRB2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5134236-A Analgesics, antidepressants, anticonvulsants HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1992-07-28 US disclosed
US-4999356-A Analgesics, antidepressants, anticonvulsants HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1991-03-12 US disclosed
EP-0302423-A2 1-Phenyl-3-(1-piperazinyl)-1h-indazoles, a process and intermediates for their preparation, and the use thereof as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1989-02-08 EP disclosed