Bromide

Bromide

SCHEMBL9682734

CCc1cc([P+](c2ccccc2)(c2ccccc2)c2ccccc2)c(=O)[nH]c1COCc1ccccc1.[Br-]

nearest known ligand 0.37

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHECHKACHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNB1CHRNDCHRNECHRNGHRH2OPRM1

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.37
HCAR2 Q8TDS4 2/20 0.36
CDK5 Q00535 2/20 0.36
CDK5R1 Q15078 2/20 0.36
ALDH1A1 P00352 4/20 0.35
PDE10A Q9Y233 2/20 0.35
TK1 P04183 1/20 0.33
DAO P14920 1/20 0.32
LMNA P02545 1/20 0.32
USP2 O75604 1/20 0.31
MAPK1 P28482 1/20 0.31
HPGD P15428 1/20 0.31
DPYD Q12882 1/20 0.31
APP P05067 1/20 0.31
MMP13 P45452 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9680279 0.77 TSHR (0.41) TSHRHCAR2CDK5CDK5R1ALDH1A1
SCHEMBL9449305 0.75 SMN1; SMN2 (0.47) TSHRHCAR2CDK5CDK5R1ALDH1A1
SCHEMBL9455953 0.74 TSHR (0.38) TSHRHCAR2CDK5CDK5R1ALDH1A1
SCHEMBL14394524 0.64 TSHR (0.62) TSHRALDH1A1DAOLMNAMAPK1
SCHEMBL28301231 0.63 TSHR (0.83) TSHRALDH1A1DAOMAPK1
Propane SCHEMBL11584021 0.63 TSHR (0.83) TSHRALDH1A1MAPK1
Benzoquinone SCHEMBL8469988 0.61 TSHR (0.71) TSHRALDH1A1DAOLMNAMAPK1
SCHEMBL20599933 0.61 TYMP (0.50) TSHRALDH1A1LMNA
SCHEMBL5311581 0.60 TSHR (1.00) TSHRALDH1A1LMNA
SCHEMBL27380 0.60 TSHR (1.00) TSHRALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0481802-A1 Hydroxylated inhibitors of HIV reverse transcriptase MERCK & CO. INC. (US) 1992-04-22 EP disclosed