SCHEMBL9684142

SCHEMBL9684142

Oc1cccc2ccc(CBr)nc12

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 2/20 0.63
METAP2 P50579 2/20 0.53
PLAU P00749 1/20 0.53
NCF1 P14598 1/20 0.53
ALOX12 P18054 2/20 0.52
ALDH1A1 P00352 1/20 0.52
CYP1A2 P05177 1/20 0.52
CYP3A4 P08684 1/20 0.52
CYP2C9 P11712 1/20 0.52
HPGD P15428 1/20 0.52
CYP2C19 P33261 1/20 0.52
HIF1A Q16665 1/20 0.52
HSD17B10 Q99714 1/20 0.52
KDM4E B2RXH2 3/20 0.49
KMT2A Q03164 3/20 0.49
SOS2 Q07890 1/20 0.49
PIM1 P11309 1/20 0.47
TSHR P16473 2/20 0.47
MMP2 P08253 1/20 0.47
CHRM1 P11229 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4393939 0.85 METAP2 (0.53) CCR1METAP2PLAUNCF1ALOX12
SCHEMBL4394002 0.84 METAP2 (0.57) CCR1METAP2PLAUNCF1ALOX12
SCHEMBL3212638 0.84 METAP2 (0.57) CCR1METAP2PLAUNCF1ALOX12
SCHEMBL9220073 0.82 CCR1 (0.65) CCR1METAP2PLAUNCF1ALOX12
SCHEMBL2522559 0.81 PLAU (0.58) CCR1METAP2PLAUNCF1ALOX12
SCHEMBL1101005 0.81 PARP1 (0.58) METAP2PLAUNCF1ALOX12ALDH1A1
SCHEMBL2781605 0.81 METAP2 (0.53) CCR1METAP2PLAUNCF1ALOX12
SCHEMBL10437729 0.80 METAP2 (0.49) CCR1METAP2PLAUNCF1ALOX12
Hydrochloric Acid SCHEMBL6535609 0.79 METAP2 (0.52) CCR1METAP2PLAUNCF1ALOX12
Hydrochloric Acid SCHEMBL1978354 0.79 PLAU (0.56) CCR1METAP2PLAUNCF1ALOX12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104994853-A Dihydro-6-azaphenalene derivatives for the treatment of cns, oncological diseases and related disorders WARNER BABCOCK INST FOR GREEN CHEMISTRY LLC 2015-10-21 CN disclosed
US-5082666-A Drugs, sweeteners LABORATOIRES BEAUFOUR (FR) 1992-01-21 US disclosed