SCHEMBL9684591

SCHEMBL9684591

O=[N+]([O-])c1cnc(N2CCNCC2)c([N+](=O)[O-])c1

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.74
HTT P42858 2/20 0.74
MAPK1 P28482 1/20 0.74
ADRB1 P08588 1/20 0.49
SIRT6 Q8N6T7 1/20 0.49
MAPT P10636 8/20 0.46
POLB P06746 1/20 0.46
RECQL P46063 1/20 0.46
CYP1A2 P05177 3/20 0.45
CYP2C19 P33261 3/20 0.45
HTR3E A5X5Y0 1/20 0.45
HTR3B O95264 1/20 0.45
CYP3A4 P08684 1/20 0.45
SLC6A4 P31645 1/20 0.45
THPO P40225 1/20 0.45
HTR3A P46098 1/20 0.45
HTR3D Q70Z44 1/20 0.45
HTR3C Q8WXA8 1/20 0.45
LMNA P02545 1/20 0.44
GAA P10253 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29046091 0.87 ALDH1A1 (0.56) ALDH1A1HTTMAPK1ADRB1SIRT6
SCHEMBL30412573 0.87 ALDH1A1 (0.56) ALDH1A1HTTMAPK1ADRB1SIRT6
SCHEMBL1093120 0.86 ALDH1A1 (0.97) ALDH1A1HTTMAPK1MAPTPOLB
SCHEMBL907889 0.85 ALDH1A1 (0.54) ALDH1A1HTTMAPK1ADRB1SIRT6
SCHEMBL4676953 0.85 ALDH1A1 (1.00) ALDH1A1HTTMAPK1MAPTPOLB
SCHEMBL4679344 0.85 ALDH1A1 (1.00) ALDH1A1HTTMAPK1MAPTPOLB
Hydrochloric Acid SCHEMBL3174215 0.84 ALDH1A1 (0.52) ALDH1A1HTTMAPK1ADRB1SIRT6
SCHEMBL899829 0.84 ALDH1A1 (0.52) ALDH1A1HTTMAPK1ADRB1SIRT6
SCHEMBL903045 0.84 ALDH1A1 (0.52) ALDH1A1HTTMAPK1ADRB1SIRT6
SCHEMBL13075786 0.84 ALDH1A1 (0.52) ALDH1A1HTTMAPK1ADRB1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0188094-B1 QUINAZOLINE DERIVATIVES AND ANTIHYPERTENSIVE PREPARATIONS CONTAINING SAME AS EFFECTIVE COMPONENTS MITSUI PETROCHEMICAL INDUSTRIES, LTD. (JP) 1992-03-18 EP disclosed
US-4734418-A Quinazoline compounds and antihypertensives MITSUI PETROCHEMICAL INDUSTRIES, LTD. (JP) 1988-03-29 US disclosed
EP-0188094-A2 Quinazoline derivatives and antihypertensive preparations containing same as effective components MITSUI PETROCHEMICAL INDUSTRIES, LTD. (JP) 1986-07-23 EP disclosed