SCHEMBL9684889

SCHEMBL9684889

COC1(N)CCN(Cc2ccccc2)CC1

nearest known ligand 0.56

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.56
HSD17B10 Q99714 1/20 0.56
SIGMAR1 Q99720 5/20 0.55
OPRL1 P41146 2/20 0.53
MC4R P32245 1/20 0.51
POLB P06746 2/20 0.51
ALDH1A1 P00352 2/20 0.51
MEN1 O00255 1/20 0.51
CYP2C9 P11712 1/20 0.51
TSHR P16473 1/20 0.51
CYP2C19 P33261 1/20 0.51
KMT2A Q03164 1/20 0.51
HIF1A Q16665 1/20 0.51
CYP2D6 P10635 3/20 0.51
LMNA P02545 1/20 0.50
ADRA2A P08913 1/20 0.49
OPRM1 P35372 1/20 0.49
ACHE P22303 1/20 0.49
CCR3 P51677 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20571573 0.83 CYP3A4 (0.59) CYP3A4HSD17B10SIGMAR1OPRL1MC4R
SCHEMBL1994180 0.81 SIGMAR1 (0.61) CYP3A4HSD17B10SIGMAR1OPRL1MC4R
SCHEMBL20571837 0.81 OPRL1 (0.54) CYP3A4HSD17B10SIGMAR1OPRL1MC4R
SCHEMBL10509216 0.80 CYP2D6 (0.54) CYP3A4HSD17B10SIGMAR1OPRL1POLB
Hydrochloric Acid SCHEMBL15608841 0.79 CYP3A4 (0.59) CYP3A4HSD17B10SIGMAR1OPRL1MC4R
Methane SCHEMBL4247840 0.79 SIGMAR1 (0.63) CYP3A4HSD17B10SIGMAR1OPRL1MC4R
SCHEMBL22050089 0.79 OPRL1 (0.55) CYP3A4HSD17B10SIGMAR1OPRL1MC4R
SCHEMBL1992310 0.78 CYP3A4 (0.57) CYP3A4HSD17B10SIGMAR1OPRL1MC4R
SCHEMBL1586467 0.78 OPRL1 (0.58) CYP3A4HSD17B10SIGMAR1OPRL1MC4R
SCHEMBL24315818 0.78 CYP3A4 (0.53) CYP3A4HSD17B10SIGMAR1OPRL1MC4R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5132311-A Prolonging cardiac action potential repolarization G. D. SEARLE & CO. (US) 1992-07-21 US disclosed