SCHEMBL9685867

SCHEMBL9685867

CSc1ccc2c(c1)C(=O)c1ccc(Br)cc1-2

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S100A4 P26447 2/20 0.57
PTPRC P08575 1/20 0.55
BCL2 P10415 6/20 0.53
MCL1 Q07820 5/20 0.53
MAOA P21397 2/20 0.39
MAOB P27338 2/20 0.39
LCK P06239 1/20 0.39
ESR1 P03372 1/20 0.38
UGT1A1 P22309 1/20 0.38
ESR2 Q92731 1/20 0.38
CYP1A2 P05177 2/20 0.37
MAPK1 P28482 2/20 0.37
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
CA4 P22748 1/20 0.37
CA7 P43166 1/20 0.37
CA9 Q16790 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
TRPV1 Q8NER1 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29036115 0.85 MCL1 (0.46) S100A4BCL2MCL1MAOAMAOB
SCHEMBL19767754 0.83 S100A4 (0.81) S100A4PTPRCBCL2MCL1MAOA
SCHEMBL9811057 0.82 ELANE (0.53) S100A4PTPRCBCL2MCL1MAOA
SCHEMBL11294862 0.80 ELANE (0.55) S100A4PTPRCBCL2MCL1MAOA
SCHEMBL16659000 0.79 S100A4 (0.90) S100A4PTPRCBCL2MCL1MAOA
SCHEMBL762135 0.79 S100A4 (0.80) S100A4PTPRCBCL2MCL1MAOA
SCHEMBL12469932 0.79 S100A4 (0.71) S100A4PTPRCBCL2MCL1MAOA
SCHEMBL29664078 0.79 S100A4 (0.80) S100A4PTPRCBCL2MCL1MAOA
SCHEMBL30363166 0.79 S100A4 (0.71) S100A4PTPRCBCL2MCL1MAOA
SCHEMBL3717374 0.79 S100A4 (0.80) S100A4PTPRCBCL2MCL1MAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5144028-A Antibiotics MERCK & CO., INC. (US) 1992-09-01 US disclosed
EP-0469844-A1 2-(9-fluorenonyl)-carbapenem MERCK & CO. INC. (US) 1992-02-05 EP disclosed
US-5025007-A 2-(9-fluorenonyl)-carbapenem antibacterial agents MERCK & CO., INC. (US) 1991-06-18 US disclosed