SCHEMBL9686470

SCHEMBL9686470

COC(=O)C1c2[nH]c3cc(Br)ccc3c2CCN1C

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPKAPK2 P49137 3/20 0.53
EGFR P00533 1/20 0.41
ABCG2 Q9UNQ0 2/20 0.41
CYP2D6 P10635 6/20 0.40
CYP3A4 P08684 4/20 0.40
MEN1 O00255 4/20 0.40
KMT2A Q03164 4/20 0.40
CYP1A2 P05177 3/20 0.40
PDE5A O76074 2/20 0.40
CYP2C9 P11712 2/20 0.40
KCNH2 Q12809 2/20 0.40
CYP2B6 P20813 1/20 0.40
PDE10A Q9Y233 1/20 0.40
ADRA2A P08913 3/20 0.38
ADRA2B P18089 3/20 0.38
ADRA2C P18825 3/20 0.38
ADRA1D P25100 3/20 0.38
ADRA1A P35348 3/20 0.38
ADRA1B P35368 3/20 0.38
HSD17B10 Q99714 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6237305 0.81 MAPKAPK2 (0.62) MAPKAPK2HTR2A
SCHEMBL6236968 0.80 MAPKAPK2 (0.81) MAPKAPK2ABCG2CYP2D6KMT2ACYP1A2
SCHEMBL6238198 0.72 MAPKAPK2 (0.63) MAPKAPK2HSD17B10KDM4ELMNAHPGD
SCHEMBL1658785 0.69 MAPKAPK2 (1.00) MAPKAPK2ABCG2KMT2AHTR2BALDH1A1
SCHEMBL12660648 0.68 MAPKAPK2 (0.55) MAPKAPK2EGFRABCG2ADRA1DADRA1A
SCHEMBL6235510 0.68 MAPKAPK2 (0.81) MAPKAPK2ABCG2CYP2D6KMT2ACYP1A2
SCHEMBL10484426 0.68 CYP19A1 (0.52) MAPKAPK2EGFRABCG2CYP2D6CYP3A4
Hydrochloric Acid SCHEMBL31036471 0.68 KDM4E (0.68) CYP2D6MEN1KMT2ACYP1A2PDE5A
SCHEMBL16433469 0.68 SIRT1 (0.60) CYP2D6MEN1KMT2AKCNH2KDM4E
SCHEMBL9687220 0.67 MAPKAPK2 (0.50) MAPKAPK2MEN1KMT2AKDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0273321-B1 7-BROMO-BETA-CARBOLINE COMPOUND AND METHOD FOR PRODUCING SAME Kawaken Fine Chemicals Co., Ltd. (JP) 1992-04-22 EP disclosed