SCHEMBL9687662

SCHEMBL9687662

O=C1COc2cc(F)ccc2N1Cc1ccccn1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.53
SCN9A Q15858 5/20 0.47
HDAC1 Q13547 1/20 0.46
HDAC8 Q9BY41 1/20 0.46
HDAC6 Q9UBN7 1/20 0.46
HDAC5 Q9UQL6 1/20 0.46
ALDH1A1 P00352 4/20 0.46
TSHR P16473 2/20 0.46
MAPT P10636 2/20 0.46
NR3C2 P08235 2/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C9 P11712 1/20 0.44
ALOX15 P16050 1/20 0.44
CHRM1 P11229 2/20 0.44
MEN1 O00255 1/20 0.44
PKM P14618 1/20 0.44
KMT2A Q03164 1/20 0.44
CHRM5 P08912 1/20 0.44
CHRM3 P20309 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9686537 0.86 BRD4 (0.53) BRD4SCN9AHDAC1HDAC8HDAC6
SCHEMBL9685790 0.83 BRD4 (0.53) BRD4SCN9AHDAC1HDAC8HDAC6
SCHEMBL9685812 0.82 BRD4 (0.51) BRD4SCN9AHDAC1HDAC8HDAC6
SCHEMBL9687134 0.82 BRD4 (0.50) BRD4SCN9AHDAC1HDAC8HDAC6
SCHEMBL19030483 0.81 BRD4 (0.57) BRD4SCN9AALDH1A1TSHRMAPT
SCHEMBL18497028 0.80 BRD4 (0.62) BRD4SCN9AHDAC1HDAC8HDAC6
SCHEMBL9687541 0.79 BRD4 (0.50) BRD4SCN9AALDH1A1TSHRMAPT
SCHEMBL9687801 0.79 BRD4 (0.57) BRD4SCN9AALDH1A1TSHRMAPT
SCHEMBL9686559 0.79 BRD4 (0.49) BRD4SCN9AHDAC1HDAC8HDAC6
Hydrochloric Acid SCHEMBL9687303 0.78 BRD4 (0.49) BRD4SCN9AHDAC1HDAC8HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0296416-B1 BENZO-ANELLATED CYCLIC COMPOUNDS NIHON BAYER AGROCHEM K.K. (JP) 1992-07-29 EP disclosed
US-5077401-A Herbicides NIHON TOKUSHU NOYAKU SEIZO K.K. (JP) 1991-12-31 US disclosed
US-4902335-A Benzo-fused cyclic compounds NIHON TOKUSHU NOYAKU SEIZO K.K. (JP) 1990-02-20 US disclosed
EP-0296416-A1 Benzo-anellated cyclic compounds NIHON BAYER AGROCHEM K.K. (JP) 1988-12-28 EP disclosed