SCHEMBL9688232

SCHEMBL9688232

Oc1ccc(OCCCCN2CCN(c3cc(N4CCCC4)nc(N4CCCC4)n3)CC2)cc1

nearest known ligand 0.52

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 5/20 0.52
CASP5 P51878 5/20 0.52
CASP4 P49662 4/20 0.52
ALDH1A1 P00352 1/20 0.52
GAA P10253 1/20 0.52
MAPT P10636 1/20 0.52
MAOB P27338 7/20 0.50
HRH3 Q9Y5N1 6/20 0.49
SIGMAR1 Q99720 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9131269 0.99 CASP1 (0.51) CASP1CASP5CASP4ALDH1A1GAA
SCHEMBL9690170 0.99 CASP1 (0.51) CASP1CASP5CASP4ALDH1A1GAA
SCHEMBL9690117 0.93 CASP1 (0.54) CASP1CASP5CASP4ALDH1A1GAA
SCHEMBL9702244 0.88 CASP1 (0.64) CASP1CASP5CASP4HRH3SIGMAR1
SCHEMBL9688206 0.87 CASP1 (0.58) CASP1CASP5CASP4MAPTMAOB
SCHEMBL9689152 0.77 CASP1 (0.58) CASP1CASP5CASP4
SCHEMBL9128566 0.77 CASP1 (0.58) CASP1CASP5CASP4
SCHEMBL9689535 0.77 CASP1 (0.58) CASP1CASP5CASP4
SCHEMBL9690413 0.77 CASP1 (0.58) CASP1CASP5CASP4
SCHEMBL9133699 0.77 CASP1 (0.58) CASP1CASP5CASP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0358676-A1 PHARMACEUTICALLY ACTIVE AMINES THE UPJOHN COMPANY (US) 1990-03-21 EP claimed
EP-0293078-A1 Pharmaceutically active amines THE UPJOHN COMPANY (US) 1988-11-30 EP claimed
WO-1988008424-A1 PHARMACEUTICALLY ACTIVE AMINES THE UPJOHN COMPANY (US) 1988-11-03 WO claimed
US-5120843-A Nervous system disorders UPJOHN (US) 1992-06-09 US disclosed
EP-0487510-A1 Pharmaceutically active amines THE UPJOHN COMPANY (US) 1992-05-27 EP disclosed
EP-0358676-A1 PHARMACEUTICALLY ACTIVE AMINES THE UPJOHN COMPANY (US) 1990-03-21 EP disclosed
WO-1988008424-A1 PHARMACEUTICALLY ACTIVE AMINES THE UPJOHN COMPANY (US) 1988-11-03 WO disclosed