SCHEMBL9688543

SCHEMBL9688543

Cc1cc(N)c(N)cc1OC(F)F

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CD44 P16070 1/20 0.38
CYP3A4 P08684 1/20 0.37
TSHR P16473 1/20 0.37
MAPK1 P28482 1/20 0.37
BACE1 P56817 15/20 0.35
CTSD P07339 1/20 0.35
BACE2 Q9Y5Z0 1/20 0.35
APP P05067 2/20 0.35
ALDH1A1 P00352 2/20 0.33
MEN1 O00255 1/20 0.33
MAPT P10636 1/20 0.33
KMT2A Q03164 1/20 0.33
POLB P06746 1/20 0.32
GAA P10253 1/20 0.32
GFER P55789 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30695911 0.86 BACE1 (0.37) CYP3A4BACE1CTSDBACE2APP
SCHEMBL10440456 0.86 BACE1 (0.37) CYP3A4BACE1CTSDBACE2APP
SCHEMBL24696890 0.86 BACE1 (0.37) CYP3A4TSHRMAPK1BACE1CTSD
Hydrochloric Acid SCHEMBL9528218 0.81 PTK2 (0.35)
SCHEMBL10497833 0.80 CD44 (0.33) CD44CYP3A4TSHRMAPK1
SCHEMBL27397784 0.78 CYP3A4 (0.38) CYP3A4TSHRMAPK1BACE1CTSD
SCHEMBL9687372 0.77 TSHR (0.44) CYP3A4TSHRMAPK1ALDH1A1MEN1
SCHEMBL26618704 0.76 POLB (0.42) CYP3A4TSHRMAPK1BACE1CTSD
SCHEMBL7815967 0.75 ALDH1A1 (0.46) CYP3A4TSHRMAPK1ALDH1A1MEN1
SCHEMBL29739519 0.75 ALDH1A1 (0.46) CYP3A4TSHRMAPK1ALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0201575-B1 NEW PICOLINE DERIVATIVES, PREPARATION PROCESS THEREOF, UTILIZATION THEREOF AND DRUGS CONTAINING THEM Byk Gulden Lomberg Chemische Fabrik GmbH (DE) 1992-08-12 EP disclosed
US-4686230-A Picoline derivative useful as gastric acid secretion inhibitors BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1987-08-11 US disclosed
EP-0201575-A1 NEW PICOLINE DERIVATIVES, PREPARATION PROCESS THEREOF, UTILIZATION THEREOF AND DRUGS CONTAINING THEM. BYK GULDEN LOMBERG CHEM FAB (DE) 1986-11-20 EP disclosed
WO-1986002646-A1 NEW PICOLINE DERIVATIVES, PREPARATION PROCESS THEREOF, UTILIZATION THEREOF AND DRUGS CONTAINING THEM BYK GULDEN LOMBERG CHEMISCHE FABRIK GESELLSCHAFT M (DE) 1986-05-09 WO disclosed