SCHEMBL9688666

SCHEMBL9688666

Nc1cccnc1N1CCN(C(=O)OCc2ccccc2)CC1.O=C(OCc1ccccc1)N1CCN(c2ncccc2[N+](=O)[O-])CC1

nearest known ligand 0.54

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 2/20 0.54
HDAC1 Q13547 1/20 0.50
ALDH1A1 P00352 5/20 0.49
MAPT P10636 4/20 0.49
CYP1A2 P05177 3/20 0.49
CYP2C9 P11712 3/20 0.49
CYP2C19 P33261 2/20 0.49
L3MBTL1 Q9Y468 1/20 0.47
LMNA P02545 1/20 0.47
MAPK1 P28482 1/20 0.46
GRIN2B Q13224 1/20 0.44
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
POLB P06746 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8922623 0.94 GRM5 (0.60) GRM5ALDH1A1MAPTCYP1A2CYP2C9
SCHEMBL8921825 0.90 HDAC1 (0.58) GRM5HDAC1CYP2C9CYP2C19GRIN2B
SCHEMBL11474488 0.79 SMN1; SMN2 (0.60) GRM5ALDH1A1MAPTCYP1A2CYP2C9
SCHEMBL3821618 0.78 MAPT (0.56) GRM5ALDH1A1MAPTCYP1A2CYP2C9
SCHEMBL4563772 0.76 CYP1A2 (0.69) GRM5ALDH1A1MAPTCYP1A2CYP2C9
SCHEMBL8713970 0.75 ALDH1A1 (0.49) GRM5ALDH1A1MAPTCYP1A2CYP2C9
SCHEMBL12190517 0.74 GRM5 (0.58) GRM5ALDH1A1MAPTCYP1A2CYP2C9
SCHEMBL3336130 0.74 CYP1A2 (0.59) GRM5ALDH1A1MAPTCYP1A2CYP2C9
SCHEMBL29741462 0.74 CYP1A2 (0.59) GRM5ALDH1A1MAPTCYP1A2CYP2C9
SCHEMBL781659 0.73 CYP1A2 (0.87) GRM5ALDH1A1MAPTCYP1A2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0507861-A1 DIAROMATIC SUBSTITUTED ANTI-AIDS COMPOUNDS. UPJOHN CO (US) 1992-10-14 EP disclosed