SCHEMBL9689165

SCHEMBL9689165

c1cnc2[nH]c(NC3CCNC3)nc2c1

nearest known ligand 0.47

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MKNK1 Q9BUB5 1/20 0.45
MKNK2 Q9HBH9 1/20 0.45
PTPN11 Q06124 2/20 0.44
BRD4 O60885 2/20 0.42
ATAD2 Q6PL18 2/20 0.42
CHEK2 O96017 2/20 0.41
CHEK1 O14757 2/20 0.41
IDH2 P48735 1/20 0.39
PRKCZ Q05513 1/20 0.39
PRKCI P41743 1/20 0.39
PIK3CA P42336 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9688928 0.99 MKNK1 (0.44) MKNK1MKNK2PTPN11BRD4ATAD2
Hydrochloric Acid SCHEMBL9690717 0.99 MKNK1 (0.44) MKNK1MKNK2PTPN11BRD4ATAD2
Bromide SCHEMBL9689909 0.99 MKNK1 (0.44) MKNK1MKNK2PTPN11BRD4ATAD2
SCHEMBL9044459 0.92 PTPN11 (0.48) MKNK1PTPN11BRD4ATAD2
SCHEMBL9535416 0.86 PIM1 (0.48) MKNK1PTPN11CHEK2PRKCZ
Hydrochloric Acid SCHEMBL9689129 0.85 PIM1 (0.47) MKNK1PTPN11CHEK2PRKCZ
SCHEMBL9690640 0.80 CHEK1 (0.52) CHEK1
Hydrochloric Acid SCHEMBL9690626 0.79 CHEK1 (0.51) CHEK1
Hydrochloric Acid SCHEMBL9691095 0.79 CHEK1 (0.51) CHEK1
SCHEMBL9534992 0.77 CDC7 (0.54) BRD4ATAD2IDH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0297661-B1 [(Bicyclic heterocyclyl)methyl and -hetero] substituted hexahydro-1H-azepines and pyrrolidines JANSSEN PHARMACEUTICA N.V. (BE) 1992-09-16 EP disclosed