SCHEMBL9689542

SCHEMBL9689542

CCCCCCC(CCC(O)N1CCNCC1)c1cc(N2CCCC2)nc(N2CCCC2)n1

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 5/20 0.46
CASP5 P51878 5/20 0.46
CASP4 P49662 4/20 0.46
HRH4 Q9H3N8 2/20 0.35
HRH1 P35367 1/20 0.34
USP2 O75604 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
GBA1 P04062 2/20 0.32
IKBKB O14920 2/20 0.32
CETP P11597 1/20 0.32
KMT5A Q9NQR1 1/20 0.30
CHUK O15111 1/20 0.30
PDGFRA P16234 1/20 0.30
EPHA3 P29320 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9689160 1.00 CASP1 (0.46) CASP1CASP5CASP4HRH4HRH1
Hydrochloric Acid SCHEMBL9690260 0.99 CASP1 (0.45) CASP1CASP5CASP4HRH4HRH1
Hydrochloric Acid SCHEMBL9689164 0.99 CASP1 (0.45) CASP1CASP5CASP4HRH4HRH1
SCHEMBL9690206 0.96 CASP1 (0.48) CASP1CASP5CASP4HRH4HRH1
Hydrochloric Acid SCHEMBL9689568 0.95 CASP1 (0.47) CASP1CASP5CASP4HRH4HRH1
SCHEMBL9688175 0.89 CASP1 (0.51) CASP1CASP5CASP4HRH4HRH1
Hydrochloric Acid SCHEMBL9690244 0.88 CASP1 (0.50) CASP1CASP5CASP4HRH4HRH1
SCHEMBL9690419 0.82 CASP1 (0.53) CASP1CASP5CASP4HRH4HRH1
Hydrochloric Acid SCHEMBL9689526 0.81 CASP1 (0.52) CASP1CASP5CASP4HRH4HRH1
SCHEMBL9688169 0.79 CASP1 (0.46) CASP1CASP5CASP4HRH4GBA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0358676-A1 PHARMACEUTICALLY ACTIVE AMINES THE UPJOHN COMPANY (US) 1990-03-21 EP claimed
EP-0293078-A1 Pharmaceutically active amines THE UPJOHN COMPANY (US) 1988-11-30 EP claimed
WO-1988008424-A1 PHARMACEUTICALLY ACTIVE AMINES THE UPJOHN COMPANY (US) 1988-11-03 WO claimed
US-5120843-A Nervous system disorders UPJOHN (US) 1992-06-09 US disclosed
EP-0487510-A1 Pharmaceutically active amines THE UPJOHN COMPANY (US) 1992-05-27 EP disclosed
EP-0358676-A1 PHARMACEUTICALLY ACTIVE AMINES THE UPJOHN COMPANY (US) 1990-03-21 EP disclosed
WO-1988008424-A1 PHARMACEUTICALLY ACTIVE AMINES THE UPJOHN COMPANY (US) 1988-11-03 WO disclosed