SCHEMBL9689580

SCHEMBL9689580

c1ccc2c(Cn3cncn3)noc2c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 8/20 0.50
LMNA P02545 2/20 0.45
CA12 O43570 1/20 0.45
CA1 P00915 1/20 0.45
CA2 P00918 1/20 0.45
CA3 P07451 1/20 0.45
CA4 P22748 1/20 0.45
CA6 P23280 1/20 0.45
MAOB P27338 1/20 0.45
CA5A P35218 1/20 0.45
CA7 P43166 1/20 0.45
CA9 Q16790 1/20 0.45
CA13 Q8N1Q1 1/20 0.45
CA14 Q9ULX7 1/20 0.45
CA5B Q9Y2D0 1/20 0.45
BRD4 O60885 1/20 0.44
ACHE P22303 2/20 0.43
SMN1; SMN2 Q16637 4/20 0.41
CYP3A4 P08684 1/20 0.41
BLM P54132 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9689669 0.82 CYP19A1 (0.53) CYP19A1LMNASMN1; SMN2KDM4E
SCHEMBL10570210 0.80 CYP19A1 (0.44) CYP19A1SMN1; SMN2KDM4E
Hydrochloric Acid SCHEMBL9688442 0.79 CYP19A1 (0.44) CYP19A1SMN1; SMN2KDM4E
Hydrochloric Acid SCHEMBL9688871 0.79 CYP19A1 (0.38) CYP19A1MAOBBRD4ACHE
Hydrochloric Acid SCHEMBL9688723 0.79 CYP19A1 (0.44) CYP19A1LMNACYP3A4HSP90AA1
Hydrochloric Acid SCHEMBL9687944 0.79 MAPT (0.49) CYP19A1LMNAACHE
Hydrochloric Acid SCHEMBL9688795 0.79 CYP19A1 (0.46) CYP19A1KDM4E
SCHEMBL14699201 0.74 KLKB1 (0.54) LMNACA12CA1CA2CA3
SCHEMBL9688353 0.73 CYP19A1 (0.52) CYP19A1LMNACA12CA1CA2
SCHEMBL30474877 0.69 ACHE (0.56) LMNACA12CA1CA2CA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0298921-B1 1,2-BENZISOXAZOLES AND 1,2-BENZISOTHIAZOLES CIBA-GEIGY AG (CH) 1992-12-23 EP disclosed
US-4957931-A ANTICONVULSANTS, TREATMENT OF EPILEPSY CIBA-GEIGY CORPORATION (US) 1990-09-18 US disclosed
US-4859691-A Certain 1,2-benzisoxazole derivatives CIBA-GEIGY CORPORATION (US) 1989-08-22 US disclosed
EP-0298921-A1 1,2-Benzisoxazoles and 1,2-benzisothiazoles CIBA-GEIGY AG (CH) 1989-01-11 EP disclosed