SCHEMBL9689618

SCHEMBL9689618

COc1ccc(CCNCc2cc(O)ccc2O)cc1OC

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.67
ALDH1A1 P00352 2/20 0.57
SMPD1 P17405 1/20 0.57
LMNA P02545 1/20 0.57
NPSR1 Q6W5P4 1/20 0.57
SLC22A1 O15245 1/20 0.57
ADRB2 P07550 1/20 0.57
CHRM2 P08172 1/20 0.57
ADRB1 P08588 1/20 0.57
CYP3A4 P08684 1/20 0.57
CHRM1 P11229 1/20 0.57
TSHR P16473 1/20 0.57
NFKB1 P19838 1/20 0.57
SLC6A4 P31645 1/20 0.57
OPRM1 P35372 1/20 0.57
SLC6A3 Q01959 1/20 0.57
HIF1A Q16665 1/20 0.57
KDM4E B2RXH2 1/20 0.56
GLA P06280 1/20 0.56
BCHE P06276 2/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9689514 0.88 CA1 (0.65) SMN1; SMN2ALDH1A1SMPD1KDM4EGLA
SCHEMBL4542599 0.87 SMN1; SMN2 (0.64) SMN1; SMN2ALDH1A1SMPD1LMNANPSR1
SCHEMBL9073446 0.82 KDM4E (0.64) SMN1; SMN2ALDH1A1ADRB2KDM4EGLA
SCHEMBL5069115 0.82 BCHE (0.76) SMN1; SMN2ALDH1A1LMNANPSR1SLC22A1
SCHEMBL7435099 0.78 ATM (0.76) SMN1; SMN2ALDH1A1SMPD1ADRB2KDM4E
Hydrochloric Acid SCHEMBL11806441 0.77 ADRB2 (0.71) ALDH1A1LMNANPSR1SLC22A1ADRB2
SCHEMBL31364604 0.77 TAAR1 (0.69) ALDH1A1LMNAADRB2CYP3A4TSHR
Hydrochloric Acid SCHEMBL11808765 0.76 ATM (0.73) SMN1; SMN2ALDH1A1ADRB2KDM4EGLA
SCHEMBL4103633 0.76 SMPD1 (0.70) SMN1; SMN2ALDH1A1SMPD1LMNAADRB2
SCHEMBL5355216 0.76 SMN1; SMN2 (0.62) SMN1; SMN2ALDH1A1LMNANPSR1SLC22A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0293078-A1 Pharmaceutically active amines THE UPJOHN COMPANY (US) 1988-11-30 EP claimed
US-5120843-A Nervous system disorders UPJOHN (US) 1992-06-09 US disclosed
EP-0487510-A1 Pharmaceutically active amines THE UPJOHN COMPANY (US) 1992-05-27 EP disclosed
EP-0358676-A1 PHARMACEUTICALLY ACTIVE AMINES THE UPJOHN COMPANY (US) 1990-03-21 EP disclosed
EP-0293078-A1 Pharmaceutically active amines THE UPJOHN COMPANY (US) 1988-11-30 EP disclosed
WO-1988008424-A1 PHARMACEUTICALLY ACTIVE AMINES THE UPJOHN COMPANY (US) 1988-11-03 WO disclosed