SCHEMBL9689622

SCHEMBL9689622

C/C(N)=C/C(=O)OCCCCCCO

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TSHR P16473 5/20 0.44
ALDH1A1 P00352 1/20 0.44
CYP3A4 P08684 1/20 0.44
ACHE P22303 6/20 0.41
APP P05067 2/20 0.40
HCAR2 Q8TDS4 3/20 0.40
ATM Q13315 1/20 0.38
MAPT P10636 1/20 0.37
RAB9A P51151 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
HPGD P15428 1/20 0.36
GAA P10253 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10923787 1.00 TSHR (0.44) TSHRALDH1A1CYP3A4ACHEAPP
SCHEMBL10919646 1.00 TSHR (0.44) TSHRALDH1A1CYP3A4ACHEAPP
SCHEMBL29182959 0.98 TSHR (0.41) TSHRALDH1A1CYP3A4ACHEAPP
SCHEMBL31531957 0.98 TSHR (0.41) TSHRALDH1A1CYP3A4ACHEAPP
Ethylene Glycol SCHEMBL11055892 0.92 TSHR (0.42) TSHRALDH1A1CYP3A4ACHEAPP
SCHEMBL11003628 0.92 TSHR (0.50) TSHRALDH1A1CYP3A4ACHEHCAR2
SCHEMBL11006969 0.92 TSHR (0.50) TSHRALDH1A1CYP3A4ACHEHCAR2
SCHEMBL11003632 0.92 TSHR (0.50) TSHRALDH1A1CYP3A4ACHEHCAR2
SCHEMBL11006987 0.92 TSHR (0.50) TSHRALDH1A1CYP3A4ACHEHCAR2
SCHEMBL759827 0.90 TSHR (0.46) TSHRALDH1A1CYP3A4HCAR2ATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0071819-B2 DIHYDROPYRIDINES WITH A POSITIVE INOTROPIC ACTIVITY, THEIR USE IN PHARMACEUTICAL PREPARATIONS, AND PROCESSES FOR THEIR PREPARATION BAYER AG (DE) 1992-06-10 EP disclosed
EP-0071819-B1 DIHYDROPYRIDINES WITH A POSITIVE INOTROPIC ACTIVITY, THEIR USE IN PHARMACEUTICAL PREPARATIONS, AND PROCESSES FOR THEIR PREPARATION BAYER AG (DE) 1987-04-22 EP disclosed
EP-0071819-A1 Dihydropyridines with a positive inotropic activity, their use in pharmaceutical preparations, and processes for their preparation BAYER AG (DE) 1983-02-16 EP disclosed