SCHEMBL9690459

SCHEMBL9690459

Cc1c(C)c2c(c(C)c1O)CCC(C)(C(=O)N1CCN(Cc3ccccc3-c3ccc(Cl)cc3)CC1)O2

nearest known ligand 0.51

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ACHE P22303 11/20 0.51
MAOB P27338 1/20 0.51
PTGS1 P23219 1/20 0.44
PTGS2 P35354 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
TSHR P16473 1/20 0.44
BCL2 P10415 4/20 0.41
BAK1 Q16611 2/20 0.41
MEN1 O00255 1/20 0.40
RAB9A P51151 1/20 0.40
KMT2A Q03164 1/20 0.40
BCHE P06276 11/20 0.40
BCL2L1 Q07817 2/20 0.40
HTR7 P34969 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10648165 0.84 USP2 (0.50) ACHEMAOBCYP3A4TSHRBCL2
SCHEMBL2059447 0.84 TSHR (0.55) ACHEMAOBPTGS1PTGS2CYP1A2
SCHEMBL9690307 0.79 PTGS1 (0.53) ACHEMAOBPTGS1PTGS2CYP1A2
SCHEMBL9690451 0.78 TSHR (0.49) ACHEMAOBPTGS1PTGS2CYP1A2
SCHEMBL15825618 0.77 CYP3A4 (0.57) ACHEMAOBPTGS1PTGS2CYP1A2
SCHEMBL22512408 0.77 CYP3A4 (0.60) ACHEMAOBPTGS1PTGS2CYP1A2
SCHEMBL10366019 0.75 MEN1 (0.51) ACHEMAOBPTGS1PTGS2CYP1A2
SCHEMBL9690175 0.75 TSHR (0.50) ACHEPTGS1PTGS2CYP1A2CYP3A4
SCHEMBL15820153 0.75 CYP3A4 (0.60) ACHEMAOBPTGS1PTGS2CYP1A2
SCHEMBL17289288 0.75 CYP3A4 (0.60) ACHEMAOBPTGS1PTGS2CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0487510-A1 Pharmaceutically active amines THE UPJOHN COMPANY (US) 1992-05-27 EP claimed
EP-0358676-A1 PHARMACEUTICALLY ACTIVE AMINES THE UPJOHN COMPANY (US) 1990-03-21 EP claimed
EP-0293078-A1 Pharmaceutically active amines THE UPJOHN COMPANY (US) 1988-11-30 EP claimed
WO-1988008424-A1 PHARMACEUTICALLY ACTIVE AMINES THE UPJOHN COMPANY (US) 1988-11-03 WO claimed
EP-0358676-A1 PHARMACEUTICALLY ACTIVE AMINES THE UPJOHN COMPANY (US) 1990-03-21 EP disclosed
WO-1988008424-A1 PHARMACEUTICALLY ACTIVE AMINES THE UPJOHN COMPANY (US) 1988-11-03 WO disclosed