SCHEMBL9693347

SCHEMBL9693347

Nc1ccc2nc3[nH]c(=O)[nH]c3cc2c1

nearest known ligand 0.67

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 20/20 0.67
PDE3A Q14432 20/20 0.67
PDE2A O00408 3/20 0.63
P2RY12 Q9H244 6/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10758549 0.80 PDE3B (1.00) PDE3BPDE3APDE2AP2RY12
SCHEMBL10757077 0.80 PDE3B (1.00) PDE3BPDE3APDE2AP2RY12
SCHEMBL10758208 0.80 PDE3B (1.00) PDE3BPDE3APDE2AP2RY12
SCHEMBL10758507 0.80 PDE3B (0.67) PDE3BPDE3APDE2AP2RY12
Water SCHEMBL10768601 0.79 PDE3B (0.97) PDE3BPDE3APDE2AP2RY12
SCHEMBL2014813 0.77 PDE3B (1.00) PDE3BPDE3APDE2AP2RY12
SCHEMBL31061086 0.77 PDE3B (1.00) PDE3BPDE3APDE2AP2RY12
SCHEMBL32659859 0.76 PDE3B (0.80) PDE3BPDE3APDE2AP2RY12
SCHEMBL10758046 0.76 PDE3B (1.00) PDE3BPDE3APDE2AP2RY12
SCHEMBL10760128 0.73 PDE3B (1.00) PDE3BPDE3APDE2AP2RY12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0252503-B1 AMINOIMIDAZOQUINOLINE DERIVATIVES Bristol-Myers Squibb Company (US) 1992-11-19 EP claimed
US-4701459-A 7-amino-1,3-dihydro-2H-imidazo[4,5-b]quinolin 2-ones and method for inhibiting phosphodiesterase and blood platelet aggregation BRISTOL-MYERS COMPANY (US) 1987-10-20 US claimed
EP-0252503-B1 AMINOIMIDAZOQUINOLINE DERIVATIVES Bristol-Myers Squibb Company (US) 1992-11-19 EP disclosed
EP-0252503-A1 Aminoimidazoquinoline derivatives Bristol-Myers Squibb Company (US) 1988-01-13 EP disclosed
US-4701459-A 7-amino-1,3-dihydro-2H-imidazo[4,5-b]quinolin 2-ones and method for inhibiting phosphodiesterase and blood platelet aggregation BRISTOL-MYERS COMPANY (US) 1987-10-20 US disclosed
US-4701459-A 7-amino-1,3-dihydro-2H-imidazo[4,5-b]quinolin 2-ones and method for inhibiting phosphodiesterase and blood platelet aggregation BRISTOL-MYERS COMPANY (US) 1987-10-20 US disclosed