SCHEMBL9694471

SCHEMBL9694471

N#Cc1cccc(C(=O)NC2CCCCNC2=O)c1

nearest known ligand 0.62

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 3/20 0.62
NPC1 O15118 2/20 0.62
KDM1A O60341 1/20 0.57
ALDH1A1 P00352 3/20 0.55
KDM4E B2RXH2 1/20 0.54
GRM5 P41594 2/20 0.51
CCR2 P41597 3/20 0.49
CHEK1 O14757 1/20 0.48
TACR2 P21452 1/20 0.45
TACR1 P25103 1/20 0.45
DDB1 Q16531 1/20 0.45
CRBN Q96SW2 1/20 0.45
LMNA P02545 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
HPGDS O60760 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8381645 0.82 RAB9A (0.75) RAB9ANPC1KDM1AALDH1A1KDM4E
SCHEMBL15087624 0.82 RAB9A (0.75) RAB9ANPC1KDM1AALDH1A1KDM4E
SCHEMBL5740526 0.81 CRBN (0.69) GRM5DDB1CRBN
SCHEMBL4999518 0.81 RAB9A (0.56) RAB9ANPC1KDM1AALDH1A1KDM4E
SCHEMBL14856587 0.80 RAB9A (0.61) RAB9ANPC1KDM1AALDH1A1KDM4E
SCHEMBL14856267 0.79 RAB9A (0.59) RAB9ANPC1KDM1AALDH1A1KDM4E
SCHEMBL14856372 0.79 RAB9A (0.59) RAB9ANPC1KDM1AALDH1A1KDM4E
SCHEMBL8312018 0.79 GRM5 (0.59) RAB9ANPC1KDM4EGRM5CHEK1
SCHEMBL26407280 0.78 RAB9A (0.69) RAB9ANPC1KDM1AKDM4EGRM5
SCHEMBL4077366 0.78 RAB9A (0.68) RAB9ANPC1KDM1AALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5118806-A Enzyme inhibitor for lipoxygenase; useful for treating cancer, hepatic diseases, inflammation, cerebrovascular diseases TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1992-06-02 US disclosed