SCHEMBL9696256

SCHEMBL9696256

C[C@@H](O)[C@H]1C(=O)N2C(C(=O)O)=C(SCSc3cccnc3)[C@H](C)[C@H]12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.43
PTGS1 P23219 1/20 0.43
PDE4A P27815 1/20 0.43
CACNA1C Q13936 1/20 0.42
ABCC2 Q92887 1/20 0.37
KDM4E B2RXH2 2/20 0.34
LMNA P02545 1/20 0.34
FAP Q12884 1/20 0.33
ELANE P08246 1/20 0.33
ALDH1A1 P00352 3/20 0.32
SMN1; SMN2 Q16637 2/20 0.31
NPC1 O15118 1/20 0.31
RAB9A P51151 1/20 0.31
ALOX15 P16050 2/20 0.31
GLA P06280 1/20 0.31
TSHR P16473 1/20 0.31
CASP1 P29466 1/20 0.31
HSD17B10 Q99714 1/20 0.31
SORT1 Q99523 1/20 0.31
HTT P42858 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9696350 0.89 ESR1 (0.47) ESR1PTGS1PDE4ACACNA1CABCC2
SCHEMBL9695363 0.88 CACNA1C (0.44) ESR1PTGS1PDE4ACACNA1CABCC2
SCHEMBL9696757 0.86 ESR1 (0.41) ESR1PTGS1PDE4ACACNA1CABCC2
SCHEMBL9741317 0.86 ESR1 (0.41) ESR1PTGS1PDE4ACACNA1CABCC2
SCHEMBL9695126 0.82 CACNA1C (0.44) ESR1PTGS1PDE4ACACNA1CABCC2
SCHEMBL9738966 0.82 CACNA1C (0.44) ESR1PTGS1PDE4ACACNA1CABCC2
SCHEMBL9696455 0.82 ESR1 (0.44) ESR1PTGS1PDE4ACACNA1CABCC2
SCHEMBL9696313 0.81 CACNA1C (0.43) ESR1PTGS1PDE4ACACNA1CABCC2
SCHEMBL9696942 0.80 CACNA1C (0.45) ESR1PTGS1PDE4ACACNA1CABCC2
SCHEMBL9696978 0.80 CACNA1C (0.45) ESR1PTGS1PDE4ACACNA1CABCC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5116833-A ANTIBIOTIC C-3 DITHIOACETAL-SUBSTITUTED CARBAPENEM COMPOUNDS, COMPOSITIONS, AND METHODS OF USE THEREOF BRISTOL-MYERS SQUIBB COMPANY (US) 1992-05-26 US claimed
EP-0481511-A2 Antibiotic C-3 dithioacetal-substituted carbapenem compounds, compositions, and use thereof Bristol-Myers Squibb Company (US) 1992-04-22 EP claimed
US-5116833-A ANTIBIOTIC C-3 DITHIOACETAL-SUBSTITUTED CARBAPENEM COMPOUNDS, COMPOSITIONS, AND METHODS OF USE THEREOF BRISTOL-MYERS SQUIBB COMPANY (US) 1992-05-26 US disclosed
EP-0481511-A2 Antibiotic C-3 dithioacetal-substituted carbapenem compounds, compositions, and use thereof Bristol-Myers Squibb Company (US) 1992-04-22 EP disclosed