SCHEMBL9696757

SCHEMBL9696757

C[C@@H](O)[C@H]1C(=O)N2C(C(=O)O)=C(SCSCc3cccnc3)[C@H](C)[C@H]12

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.41
PTGS1 P23219 1/20 0.41
PDE4A P27815 1/20 0.41
CACNA1C Q13936 1/20 0.40
ABCC2 Q92887 1/20 0.36
TBXAS1 P24557 2/20 0.35
ALDH1A1 P00352 2/20 0.35
ELANE P08246 1/20 0.35
PKM P14618 1/20 0.34
DAO P14920 1/20 0.33
LMNA P02545 1/20 0.33
TP53 P04637 1/20 0.33
KDM4E B2RXH2 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33
HPGD P15428 1/20 0.33
ALOX15 P16050 1/20 0.33
HSD17B10 Q99714 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9741317 1.00 ESR1 (0.41) ESR1PTGS1PDE4ACACNA1CABCC2
SCHEMBL9696446 0.90 ESR1 (0.45) ESR1PTGS1PDE4ACACNA1CABCC2
SCHEMBL9696790 0.89 ELANE (0.37) ESR1PTGS1PDE4ACACNA1CTBXAS1
SCHEMBL9696256 0.86 ESR1 (0.43) ESR1PTGS1PDE4ACACNA1CABCC2
SCHEMBL10440557 0.84 TBXAS1 (0.39) ESR1PTGS1PDE4ACACNA1CTBXAS1
SCHEMBL9695348 0.83 ESR1 (0.42) ESR1PTGS1PDE4ACACNA1CABCC2
SCHEMBL9696273 0.82 ELANE (0.40) ALDH1A1ELANEPKMKDM4E
SCHEMBL21081301 0.81 ESR1 (0.48) ESR1PTGS1PDE4ACACNA1CABCC2
SCHEMBL10440288 0.81 ESR1 (0.48) ESR1PTGS1PDE4ACACNA1CABCC2
SCHEMBL9695363 0.80 CACNA1C (0.44) ESR1PTGS1PDE4ACACNA1CABCC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5116833-A ANTIBIOTIC C-3 DITHIOACETAL-SUBSTITUTED CARBAPENEM COMPOUNDS, COMPOSITIONS, AND METHODS OF USE THEREOF BRISTOL-MYERS SQUIBB COMPANY (US) 1992-05-26 US claimed
EP-0481511-A2 Antibiotic C-3 dithioacetal-substituted carbapenem compounds, compositions, and use thereof Bristol-Myers Squibb Company (US) 1992-04-22 EP claimed
US-5116833-A ANTIBIOTIC C-3 DITHIOACETAL-SUBSTITUTED CARBAPENEM COMPOUNDS, COMPOSITIONS, AND METHODS OF USE THEREOF BRISTOL-MYERS SQUIBB COMPANY (US) 1992-05-26 US disclosed
EP-0481511-A2 Antibiotic C-3 dithioacetal-substituted carbapenem compounds, compositions, and use thereof Bristol-Myers Squibb Company (US) 1992-04-22 EP disclosed