SCHEMBL9699279

SCHEMBL9699279

COc1ccc(C(=O)c2c(C)n3c4c(cc(OC)cc24)OCC3CN)cc1

nearest known ligand 0.59

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 6/20 0.45
CNR2 P34972 5/20 0.45
CYP3A4 P08684 2/20 0.45
MEN1 O00255 1/20 0.45
CYP2C9 P11712 1/20 0.45
KMT2A Q03164 1/20 0.45
POLB P06746 1/20 0.39
GAA P10253 1/20 0.39
ALDH1A1 P00352 3/20 0.39
TP53 P04637 1/20 0.39
CYP1A2 P05177 1/20 0.39
TSHR P16473 1/20 0.39
RECQL P46063 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
MAPT P10636 1/20 0.39
NPC1 O15118 1/20 0.39
MTOR P42345 1/20 0.39
RAB9A P51151 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9699327 0.91 CNR1 (0.43) CNR1CNR2CYP3A4MEN1CYP2C9
SCHEMBL9700377 0.88 CNR1 (0.44) CNR1CNR2CYP3A4MEN1CYP2C9
SCHEMBL9700289 0.87 CNR1 (0.54) CNR1CNR2CYP3A4MEN1CYP2C9
SCHEMBL9700269 0.87 CNR1 (0.54) CNR1CNR2CYP3A4MEN1CYP2C9
SCHEMBL9700352 0.86 CNR1 (0.52) CNR1CNR2CYP3A4MEN1CYP2C9
SCHEMBL9701369 0.85 CNR1 (0.51) CNR1CNR2CYP3A4MEN1CYP2C9
SCHEMBL9700104 0.82 CNR1 (0.49) CNR1CNR2CYP3A4MEN1CYP2C9
SCHEMBL9700097 0.81 CNR1 (0.39) CNR1CNR2CYP3A4MEN1CYP2C9
SCHEMBL9728704 0.80 CNR1 (0.42) CNR1CNR2CYP3A4MEN1CYP2C9
SCHEMBL9701388 0.79 CNR1 (0.51) CNR1CNR2CYP3A4MEN1CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5112820-A Vision defects STERLING DRUG INC. (US) 1992-05-12 US disclosed
US-5109135-A 2- or 3-aminomethyl-4-amino-3,4-dihydro-2H-1,4-benzoxazine intermediates STERLING DRUG INC. (US) 1992-04-28 US disclosed
US-5066803-A Chemical intermediates for analgesics STERLING DRUG INC. (US) 1991-11-19 US disclosed
US-4939138-A 2- and 3-aminomethyl-6-arylcarbonyl-2,3-dihydropyrrolo(1,2,3-DE)-1,4-benzoxazines STERLING DRUG INC. (US) 1990-07-03 US disclosed