SCHEMBL9728704

SCHEMBL9728704

CNCC1COc2cc(Cl)cc3c(C(=O)c4ccc(OC)cc4)c(C)n1c23

nearest known ligand 0.55

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 3/20 0.42
CNR2 P34972 2/20 0.42
MEN1 O00255 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2C9 P11712 1/20 0.42
KMT2A Q03164 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.39
POLB P06746 1/20 0.38
GAA P10253 1/20 0.38
TP53 P04637 1/20 0.37
MAPT P10636 1/20 0.36
RAB9A P51151 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9700377 0.92 CNR1 (0.44) CNR1CNR2MEN1CYP3A4CYP2C9
SCHEMBL9699327 0.89 CNR1 (0.43) CNR1CNR2MEN1CYP3A4CYP2C9
SCHEMBL9700318 0.86 CNR1 (0.51) CNR1CNR2MEN1CYP3A4CYP2C9
SCHEMBL9701388 0.86 CNR1 (0.51) CNR1CNR2MEN1CYP3A4CYP2C9
SCHEMBL9700267 0.85 CNR1 (0.50) CNR1CNR2MEN1CYP3A4CYP2C9
SCHEMBL9701647 0.84 CNR1 (0.49) CNR1CNR2MEN1CYP3A4CYP2C9
SCHEMBL9699353 0.81 CNR1 (0.47) CNR1CNR2MEN1CYP3A4CYP2C9
SCHEMBL9699345 0.80 CNR1 (0.38) CNR1CNR2MEN1CYP3A4CYP2C9
SCHEMBL9699279 0.80 CNR1 (0.45) CNR1CNR2MEN1CYP3A4CYP2C9
SCHEMBL9700269 0.78 CNR1 (0.54) CNR1CNR2MEN1CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5109135-A 2- or 3-aminomethyl-4-amino-3,4-dihydro-2H-1,4-benzoxazine intermediates STERLING DRUG INC. (US) 1992-04-28 US disclosed
US-5066803-A Chemical intermediates for analgesics STERLING DRUG INC. (US) 1991-11-19 US disclosed
WO-1990007505-A1 2- AND 3-AMINOMETHYL-6-ARYLCARBONYL-2,3-DIHYDROPYRROLO[1,2,3-de]-1,4-BENZOXAZINES STERLING DRUG INC. (US) 1990-07-12 WO disclosed