SCHEMBL9700129

SCHEMBL9700129

Cc1c(Sc2ccccc2)c2cc(Cl)cc3c2n1C(CN1CCN(C)CC1)CO3

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 5/20 0.38
CNR2 P34972 5/20 0.38
CYP3A4 P08684 2/20 0.38
CYP2C9 P11712 2/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
HTR1A P08908 2/20 0.37
DRD2 P14416 2/20 0.37
DRD4 P21917 2/20 0.37
ALDH1A1 P00352 3/20 0.37
MAPT P10636 1/20 0.37
NPC1 O15118 1/20 0.37
MTOR P42345 1/20 0.37
RAB9A P51151 1/20 0.37
RGS12 O14924 1/20 0.35
GMNN O75496 1/20 0.35
LMNA P02545 1/20 0.35
TP53 P04637 1/20 0.35
CYP2D6 P10635 1/20 0.35
ALOX15 P16050 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9701429 0.92 CNR1 (0.39) CNR1CNR2CYP3A4CYP2C9MEN1
SCHEMBL9701305 0.92 CNR1 (0.39) CNR1CNR2CYP3A4CYP2C9MEN1
SCHEMBL9728392 0.90 CNR1 (0.38) CNR1CNR2CYP3A4CYP2C9MEN1
SCHEMBL9700297 0.87 CNR1 (0.36) CNR1CNR2CYP3A4CYP2C9MEN1
SCHEMBL9699362 0.87 CNR1 (0.39) CNR1CNR2CYP3A4CYP2C9MEN1
SCHEMBL9701684 0.87 CNR1 (0.36) CNR1CNR2CYP3A4CYP2C9MEN1
SCHEMBL9700286 0.85 PTGDR2 (0.34) CNR1CNR2CYP3A4CYP2C9MEN1
SCHEMBL9701576 0.83 PTGDR2 (0.33) CNR1CNR2CYP3A4CYP2C9MEN1
SCHEMBL9701551 0.79 CNR1 (0.40) CNR1CNR2CYP3A4CYP2C9MEN1
SCHEMBL9700330 0.79 CNR1 (0.40) CNR1CNR2CYP3A4CYP2C9MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5112820-A Vision defects STERLING DRUG INC. (US) 1992-05-12 US disclosed
US-5109135-A 2- or 3-aminomethyl-4-amino-3,4-dihydro-2H-1,4-benzoxazine intermediates STERLING DRUG INC. (US) 1992-04-28 US disclosed
US-5066803-A Chemical intermediates for analgesics STERLING DRUG INC. (US) 1991-11-19 US disclosed
WO-1990007505-A1 2- AND 3-AMINOMETHYL-6-ARYLCARBONYL-2,3-DIHYDROPYRROLO[1,2,3-de]-1,4-BENZOXAZINES STERLING DRUG INC. (US) 1990-07-12 WO disclosed
US-4939138-A 2- and 3-aminomethyl-6-arylcarbonyl-2,3-dihydropyrrolo(1,2,3-DE)-1,4-benzoxazines STERLING DRUG INC. (US) 1990-07-03 US disclosed