SCHEMBL9701576

SCHEMBL9701576

CNCC1COc2cc(Cl)cc3c(Sc4ccccc4)c(C)n1c23

nearest known ligand 0.33

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 7/20 0.33
AKR1B1 P15121 5/20 0.33
CNR1 P21554 4/20 0.31
CNR2 P34972 4/20 0.31
MEN1 O00255 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2C9 P11712 1/20 0.31
KMT2A Q03164 1/20 0.31
ENPP2 Q13822 1/20 0.30
CYP2D6 P10635 2/20 0.30
SLC6A2 P23975 2/20 0.30
SLC6A4 P31645 2/20 0.30
ALDH1A1 P00352 2/20 0.30
HTR6 P50406 1/20 0.30
MAPT P10636 1/20 0.30
NPC1 O15118 1/20 0.30
MTOR P42345 1/20 0.30
RAB9A P51151 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9700286 0.88 PTGDR2 (0.34) PTGDR2AKR1B1CNR1CNR2MEN1
SCHEMBL9700074 0.86 TUBB4A (0.33) PTGDR2AKR1B1CNR1CNR2MEN1
SCHEMBL9701305 0.85 CNR1 (0.39) PTGDR2AKR1B1CNR1CNR2MEN1
SCHEMBL9701429 0.85 CNR1 (0.39) PTGDR2AKR1B1CNR1CNR2MEN1
SCHEMBL9700129 0.83 CNR1 (0.38) CNR1CNR2MEN1CYP3A4CYP2C9
SCHEMBL9728392 0.83 CNR1 (0.38) PTGDR2AKR1B1CNR1CNR2MEN1
SCHEMBL9700297 0.81 CNR1 (0.36) CNR1CNR2MEN1CYP3A4CYP2C9
SCHEMBL9701684 0.80 CNR1 (0.36) CNR1CNR2MEN1CYP3A4CYP2C9
SCHEMBL9701680 0.79
SCHEMBL9700412 0.74 DRD2 (0.33) PTGDR2AKR1B1CNR1CNR2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5112820-A Vision defects STERLING DRUG INC. (US) 1992-05-12 US disclosed
US-5109135-A 2- or 3-aminomethyl-4-amino-3,4-dihydro-2H-1,4-benzoxazine intermediates STERLING DRUG INC. (US) 1992-04-28 US disclosed
US-5066803-A Chemical intermediates for analgesics STERLING DRUG INC. (US) 1991-11-19 US disclosed
WO-1990007505-A1 2- AND 3-AMINOMETHYL-6-ARYLCARBONYL-2,3-DIHYDROPYRROLO[1,2,3-de]-1,4-BENZOXAZINES STERLING DRUG INC. (US) 1990-07-12 WO disclosed
US-4939138-A 2- and 3-aminomethyl-6-arylcarbonyl-2,3-dihydropyrrolo(1,2,3-DE)-1,4-benzoxazines STERLING DRUG INC. (US) 1990-07-03 US disclosed