SCHEMBL9700386

SCHEMBL9700386

CC(=O)CC(=O)c1ccc(C)cc1S

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 5/20 0.46
NPC1 O15118 3/20 0.46
IDO1 P14902 2/20 0.41
TDO2 P48775 2/20 0.41
KDM4E B2RXH2 3/20 0.39
HPGD P15428 3/20 0.39
HTT P42858 3/20 0.39
SMN1; SMN2 Q16637 3/20 0.39
LMNA P02545 2/20 0.39
MAPT P10636 2/20 0.39
NPSR1 Q6W5P4 2/20 0.39
KCNH2 Q12809 1/20 0.39
KMT2A Q03164 5/20 0.39
MEN1 O00255 4/20 0.39
POLB P06746 1/20 0.39
TDP1 Q9NUW8 1/20 0.37
PLG P00747 2/20 0.37
KLK1 P06870 2/20 0.37
KLK6 Q92876 2/20 0.37
TAS1R3 Q7RTX0 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9274995 0.81 RAB9A (0.53) RAB9ANPC1IDO1TDO2HTT
SCHEMBL8464964 0.80 RAB9A (0.70) RAB9ANPC1IDO1TDO2KDM4E
SCHEMBL31320843 0.80 RAB9A (0.70) RAB9ANPC1IDO1TDO2KDM4E
SCHEMBL11332571 0.80 GSK3B (0.50) RAB9ANPC1IDO1TDO2HPGD
SCHEMBL9700314 0.79 RAB9A (0.41) RAB9ANPC1IDO1TDO2KDM4E
SCHEMBL11165907 0.79 CYP2A6 (0.42) RAB9ANPC1KDM4EHPGDSMN1; SMN2
SCHEMBL9274950 0.78 MEN1 (0.61) RAB9ANPC1KDM4EHTTSMN1; SMN2
SCHEMBL4187193 0.76 RAB9A (0.62) RAB9ANPC1IDO1TDO2KDM4E
P-Xylene SCHEMBL11798546 0.76 MEN1 (0.59) RAB9ANPC1KDM4EHTTSMN1; SMN2
SCHEMBL8611741 0.76 MAPT (0.52) NPC1KDM4EHPGDHTTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5112820-A Vision defects STERLING DRUG INC. (US) 1992-05-12 US disclosed
US-5109135-A 2- or 3-aminomethyl-4-amino-3,4-dihydro-2H-1,4-benzoxazine intermediates STERLING DRUG INC. (US) 1992-04-28 US disclosed
US-5066803-A Chemical intermediates for analgesics STERLING DRUG INC. (US) 1991-11-19 US disclosed
WO-1990007505-A1 2- AND 3-AMINOMETHYL-6-ARYLCARBONYL-2,3-DIHYDROPYRROLO[1,2,3-de]-1,4-BENZOXAZINES STERLING DRUG INC. (US) 1990-07-12 WO disclosed
US-4939138-A 2- and 3-aminomethyl-6-arylcarbonyl-2,3-dihydropyrrolo(1,2,3-DE)-1,4-benzoxazines STERLING DRUG INC. (US) 1990-07-03 US disclosed