SCHEMBL9700561

SCHEMBL9700561

O=C(O)C(O)(C(=O)c1ccccc1)C(O)(C(=O)O)C(=O)c1ccccc1.c1ccc2c(c1)NC(CN1CCOCC1)CO2

nearest known ligand 0.71

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.71
ALDH1A1 P00352 7/20 0.41
MAPT P10636 4/20 0.41
KMT2A Q03164 3/20 0.41
CYP3A4 P08684 2/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C19 P33261 1/20 0.37
CNR1 P21554 4/20 0.36
CNR2 P34972 4/20 0.36
MEN1 O00255 1/20 0.36
CYP2C9 P11712 1/20 0.36
LMNA P02545 2/20 0.36
RAB9A P51151 2/20 0.36
HTT P42858 1/20 0.36
ATM Q13315 1/20 0.36
HIF1A Q16665 1/20 0.36
KDM4E B2RXH2 1/20 0.36
NPC1 O15118 1/20 0.35
MTOR P42345 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9701340 0.84 GAA (1.00) GAAALDH1A1KMT2ACYP3A4CYP2D6
SCHEMBL9700564 0.81 GAA (0.67) GAAALDH1A1MAPTKMT2ACYP2D6
SCHEMBL9701616 0.73 GAA (0.77) GAAALDH1A1LMNA
SCHEMBL6782573 0.72 GAA (0.60) GAAALDH1A1KMT2ACNR1
SCHEMBL7298355 0.68 GAA (0.52) GAAALDH1A1MAPTKMT2AMEN1
SCHEMBL6786225 0.68 GAA (0.67) GAACYP2D6HTT
Tetrahydrofuran SCHEMBL29274508 0.66 CES1 (0.44) GAAALDH1A1MAPTKMT2ACYP2C9
SCHEMBL11555342 0.65 GAA (0.59) GAAALDH1A1RAB9AKDM4E
SCHEMBL11327486 0.65 GAA (0.57) GAAMAPTKMT2AMEN1LMNA
SCHEMBL5466546 0.65 GAA (0.57) GAAALDH1A1MAPTKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5112820-A Vision defects STERLING DRUG INC. (US) 1992-05-12 US disclosed
US-5109135-A 2- or 3-aminomethyl-4-amino-3,4-dihydro-2H-1,4-benzoxazine intermediates STERLING DRUG INC. (US) 1992-04-28 US disclosed
US-5066803-A Chemical intermediates for analgesics STERLING DRUG INC. (US) 1991-11-19 US disclosed
WO-1990007505-A1 2- AND 3-AMINOMETHYL-6-ARYLCARBONYL-2,3-DIHYDROPYRROLO[1,2,3-de]-1,4-BENZOXAZINES STERLING DRUG INC. (US) 1990-07-12 WO disclosed
US-4939138-A 2- and 3-aminomethyl-6-arylcarbonyl-2,3-dihydropyrrolo(1,2,3-DE)-1,4-benzoxazines STERLING DRUG INC. (US) 1990-07-03 US disclosed