SCHEMBL9700564

SCHEMBL9700564

O=C(OC(C(=O)O)C(OC(=O)c1ccccc1)C(=O)O)c1ccccc1.c1ccc2c(c1)NC(CN1CCOCC1)CO2

nearest known ligand 0.67

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.67
NPC1 O15118 2/20 0.46
TP53 P04637 1/20 0.42
TSHR P16473 1/20 0.42
ALDH1A1 P00352 6/20 0.41
MAPT P10636 3/20 0.39
KMT2A Q03164 2/20 0.39
L3MBTL1 Q9Y468 4/20 0.38
KDM4E B2RXH2 1/20 0.38
ALOX12 P18054 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
LMNA P02545 2/20 0.36
HTT P42858 2/20 0.36
RAB9A P51151 2/20 0.36
CYP2D6 P10635 1/20 0.36
ATM Q13315 1/20 0.36
HIF1A Q16665 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9701340 0.82 GAA (1.00) GAAALDH1A1KMT2ACYP2D6
SCHEMBL9700561 0.81 GAA (0.71) GAANPC1ALDH1A1MAPTKMT2A
SCHEMBL9701616 0.71 GAA (0.77) GAAALDH1A1LMNA
SCHEMBL6782573 0.70 GAA (0.60) GAATSHRALDH1A1KMT2A
SCHEMBL7298355 0.69 GAA (0.52) GAANPC1TP53ALDH1A1MAPT
SCHEMBL17479013 0.66 NPC1 (0.46) GAANPC1ALDH1A1MAPTKMT2A
SCHEMBL6786225 0.66 GAA (0.67) GAAHTTCYP2D6
SCHEMBL223030 0.65 TSHR (1.00) NPC1TP53TSHRALDH1A1MAPT
SCHEMBL670257 0.65 TSHR (1.00) NPC1TP53TSHRALDH1A1MAPT
SCHEMBL11886503 0.65 TSHR (1.00) NPC1TP53TSHRALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5112820-A Vision defects STERLING DRUG INC. (US) 1992-05-12 US disclosed
US-5109135-A 2- or 3-aminomethyl-4-amino-3,4-dihydro-2H-1,4-benzoxazine intermediates STERLING DRUG INC. (US) 1992-04-28 US disclosed
US-5066803-A Chemical intermediates for analgesics STERLING DRUG INC. (US) 1991-11-19 US disclosed
WO-1990007505-A1 2- AND 3-AMINOMETHYL-6-ARYLCARBONYL-2,3-DIHYDROPYRROLO[1,2,3-de]-1,4-BENZOXAZINES STERLING DRUG INC. (US) 1990-07-12 WO disclosed
US-4939138-A 2- and 3-aminomethyl-6-arylcarbonyl-2,3-dihydropyrrolo(1,2,3-DE)-1,4-benzoxazines STERLING DRUG INC. (US) 1990-07-03 US disclosed